PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 781 Products and Services

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OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

(-)-CGP-12177, [5,7-3H]-, 25µCi (925kBq)

25 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 488.00 USD

(-)-CGP-12177, [5,7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 1191.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3850.00 USD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2013.00 USD

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 1641.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 1640.00 USD
PerkinElmer

PDE Substrate iFL-cGMP, for LabChip EZ Reader

Fluorescently-labelled cGMP for Phosphodiesterase Assays (Enyzme inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
List Price : 1685.00 USD
Receptor-expressing cell lines

ValiScreen Melanocortin MC3 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Neuropeptide NPFF2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuropeptide NPFF2 receptor, in CHO-K1 cells.
List Price : 866.00 USD
Receptor-expressing cell lines

ValiScreen Galanin Gal2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Melanocortin MC4 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

ProfilerPro Kinase Peptide Substrate 13, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 13 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD

α-Bungarotoxin, [125I]-Tyr54-, 500µCi (18.5MBq)

α-bungarotoxin extracted from venom of the Taiwanese banded krait (Bungarus multicinctus) binds the nicotinic acetylcholine receptor found at the neuromuscular junction and the 7 nicotinic acetylcholine receptor in the brain.
List Price : 2106.00 USD

MK-801, (+)-[3-3H]-, 1mCi (37MBq)

1 mCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 4338.00 USD
PerkinElmer
List Price : 1159.00 USD

SDF-1α (human, recombinant), [125I]-, 5µCi

NEX346 SDF-1 a acts at the CXCR4 (fusin or LESTR) receptor. 125I-SDF-1 a competes with SDF-1 a in CXCR4 receptor binding assays.
List Price : 708.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 11, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 11 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
Price Range : 15300.00 USD - 24400.00 USD

Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 2838.00 USD

MELATONIN, [0-METHYL-3H]

250 µCi quantities of [0-METHYL-3H]-MELATONIN are available for your research.
List Price : 2184.00 USD
Receptor-expressing cell lines

Opioid Mu (OP3) (human) ValiScreen cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

WGA-PEI TYPE A PS 50 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based scintillation assays.
List Price : 39.00 USD

MK-801, (+)-[3-3H]-%, 25µCi (925kBq)

25 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 618.00 USD
Receptor-expressing cell lines

ValiScreen Angiotensin AT2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Melanocortin MC3 (mouse) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

SDF-1α (human, recombinant), [125I]-, 25µCi

NEX346 SDF-1 a acts at the CXCR4 (fusin or LESTR) receptor. 125I-SDF-1 a competes with SDF-1 a in CXCR4 receptor binding assays.
List Price : 1903.00 USD
PerkinElmer

Membrane Target Systems: hERG K+ Channel membrane preparation

Cell membranes prepared from cells stably-transfected with hERG K+ receptor, in HEK-293 cells.
List Price : 891.00 USD

Thyroxine, ([125I]-T4), L-[125I]-, 500µCi (18.5MBq), Specific Activity: 135-165µCi (5.00-6.11MBq)/µg

NEX111 L-3,5-Diiodothyronine is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1730.00 USD

Norepinephrine, Levo-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.
List Price : 1138.00 USD
PerkinElmer

Membrane Target Systems: Cannabinoid CB2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Cannabinoid CB2 receptor, in HEK-293 cells.
List Price : 891.00 USD

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 250µCi (9.25MBq)

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]- will now be made available on a fresh lot schedule. NET876100UC and NET876250UC will be available as a fresh lot once a year on March 15 in 2017.

U-69,593, [Phenyl-3,4-3H]-, 25µCi (925kBq)

25 µCi quantities of [Phenyl-3, 4-3H]-U-69,593 are available for your research.
List Price : 658.00 USD

SCH 23390, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.
List Price : 496.00 USD
Receptor-expressing cell lines

Chemokine CCR1 ValiScreen Cell Line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Prostanoid FP (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

[125I]- Epidermal Growth Factor (h, r), 5 µCi

NEX428 Epidermal Growth Factor is radioiodinated with no carrier added 125I using a lactoperoxidase procedure and is purified by reversed phase HPLC.
List Price : 690.00 USD
Receptor-expressing cell lines

ValiScreen Free Fatty Acid FFA1 (GPR40) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

CP 55940, [Side Chain-2,3,4-3H(N)]-, 25µCi (925kBq)

25 µCi quantities of [Side Chain-2, 3, 4-3H(N)]-CP 55940 are available for your research.
List Price : 637.00 USD

Amino-3-Hydroxy-5-Methylisoxazole-4-Propionic Acid (AMPA), DL-α-[5-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of DL-α-[5-Methyl-3H]- Amino-3-Hydroxy-5-Methylisoxazole-4-Propionic Acid (AMPA) are available for your research.
List Price : 540.00 USD
PerkinElmer

WGA PS Imaging Beads 500 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based scintillation assays.
List Price : 387.00 USD

Quinpirole, [N-Propyl-3H]-, 25µCi (925kBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 554.00 USD
PerkinElmer

Membrane Target Systems: Dopamine D42 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Dopamine D42 (human) receptor, in CHO-K1 cells.
List Price : 933.00 USD

"Receptor Ligand Binding" 1-50 of 781 Products and Services

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