PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 765 Products and Services

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OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

MIP-1α (human, recombinant), [125I], 25µCi

NEX298 [125I]-MIP-1α is useful in RIA, receptor studies and crosslinking experiments in the research into immune regulation.
List Price : 2318.00 USD
PerkinElmer

Membrane Target Systems: Chemokine CX3CR1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1908.00 USD

Spiperone (Spiroperidol), [Benzene ring-3H]-, 1mCi (37MBq)

1 mCi quantities of [Benzene ring-3H]-Spiperone (Spiroperidol) are available for your research.
List Price : 3367.00 USD
PerkinElmer

Membrane Target Systems: Nicotinic membrane preparation

Cell membranes prepared from IMR32 cells containing human endogenous Nicotinic receptor.
List Price : 891.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3850.00 USD
Receptor-expressing cell lines

ValiScreen Neurokinin NK2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Galanin Gal2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
Receptor-expressing cell lines

ValiScreen Purinergic P2Y6 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-5A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

SPA Imaging Select-a-Bead Kit, 6 X 500 MG

SPA bead selection kit containing beads for receptor binding studies (contains 500 mg of WGA PS, WGA YOx, WGA PEI type A, WGA PEI type B, PEI PS and poly-L-lysine beads)
List Price : 387.00 USD

Nicotine, L-(-)-[N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 466.00 USD
PerkinElmer

RNA Binding Beads (YSI) 500 MG

Uncoated SPA beads that interact with primary phosphate groups in nucleotides (oligos, DNA and RNA); membranes can also bind.
List Price : 776.00 USD

Dihydroxyphenylethylamine, 3,4-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 3, 4-[7-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 616.00 USD
List Price : 1046.00 USD
PerkinElmer

Membrane Target Systems: Histamine H3 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 6, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 6 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD

[125I]- Epidermal Growth Factor (h, r), 25 µCi

NEX428 Epidermal Growth Factor is radioiodinated with no carrier added 125I using a lactoperoxidase procedure and is purified by reversed phase HPLC.
List Price : 1523.00 USD
Receptor-expressing cell lines

cAMPZen FroZen cells, Prostanoid EP2, Human Recombinant, HEK293

Our frozen, irradiated cAMPZen cells express a variety of GPCRs for binding and functional assays. No cell culture is required prior to testing.
List Price : 506.00 USD

Ryanodine, [9,21-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [9,21-3H(N)]-Ryanodine are available for your research.
List Price : 1913.00 USD

Sauvagine, [125I]-Tyr0], 10µCi

NEX306 [125I]Tyr0-Sauvagine has been shown to be active in receptor binding assays and has been used for receptor autoradiography.
List Price : 992.00 USD
PerkinElmer

Membrane Target Systems: Neurokinin NK2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Dihydroxyphenylethylamine (Dopamine), 3,4-[Ring-2,5,6-3H]-, 1mCi (37MBq)

1 mCi quantities of 3, 4-[Ring-2, 5, 6-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 1388.00 USD
List Price : 3312.00 USD
Receptor-expressing cell lines

ValiScreen Cannabinoid CB2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Nicotine, L-(-)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 3598.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 20, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 20 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD

Diltiazem, cis-(+)-[N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of cis-(+)-[N-Methyl-3H]-Diltiazem are available for your research.
List Price : 1489.00 USD
List Price : 2120.00 USD
Receptor-expressing cell lines

ValiScreen Vasopressin V1b (rat) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 2838.00 USD
PerkinElmer

Membrane Target Systems: Orexin OX1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Ring, Methylenes-3H(N)]-Histamine Dihydrochloride are available for your research.
List Price : 1807.00 USD

Spiperone (Spiroperidol), [Benzene ring-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Benzene ring-3H]-Spiperone (Spiroperidol) are available for your research.
List Price : 1559.00 USD
List Price : 1633.00 USD

Iodoaminopotentidine, [125I], 25 µCi

NEX431 [125I]-Aminopotentidine has been shown to work in receptor binding and autoradiography and is an antagonist for histamine (H2) receptors.
List Price : 1839.00 USD

IL-6 (human, recombinant), [125I], 25µCi

NEX269 Interleukin-6 (IL-6) is a protein that in humans is encoded by the IL6 gene. IL-6 is an interleukin that acts as both a pro-inflammatory and anti-inflammatory cytokine. It is secreted by T cells and macrophages to stimulate immune response to trauma, especially burns or other tissue damage leading to inflammation.
List Price : 3924.00 USD

Scopolamine Methyl Chloride, [N-methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of [N-Methyl-3H]-Scopolamine Methyl Chloride are available for your research.
List Price : 3302.00 USD
PerkinElmer

Membrane Target Systems: Serotonin 5HT-2B (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Thyroxine, ([125I]-T4), L-[125I]-, 250µCi (9.25MBq), Specific Activity: 135-165µCi (5.00-6.11MBq)/µg

NEX111 L-3,5-Diiodothyronine is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 925.00 USD

Astemizole, [O-Methyl-3H]-, 25µCi (925kBq)

Astemizole, [O-Methyl-3H]- will now be made available on a fresh lot schedule. NET1140025UC, NET1140250UC, and NET1140001MC will be available as a fresh lot twice a year on March 6 and August 7 in 2017.
List Price : 667.00 USD

Iodo-Melatonin, 2-[125I], 50µCi

NEX236 2-[125I]-iodomelatonin has been used to identify, characterize and localize melatonin binding sites in the brain and peripheral tissues.
List Price : 941.00 USD

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