PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 756 Products and Services

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LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.
PerkinElmer

PEI - YSI Beads, 500 MG

PEI-coated SPA beads, for use in scintillation proximity assays.
List Price : 773.00 USD
List Price : 957.00 USD
PerkinElmer

Streptavidin YOX Imaging 25 X 500 MG

Streptavidin-coated SPA beads, for capturing biotinylated molecules in proximity-based scintillation assays.
List Price : 32200.00 USD

Apamin [125I]His18-NH2, 50µCi

NEX242 [125I]-Apamin is a K+ channel antagonist and can be used in the detection and quantification of K+ channel receptors. [125I]-Apamin has been used in receptor binding assays and in autoradiography.
List Price : 1415.00 USD

Glucagon, Receptor Grade, [125I]-, 50µCi

NEX207 Glucagon is radioiodinated with no carrier added 125I by a lactoperoxidase procedure and is purified by reversed phase HPLC. [125I]-Glucagon consists of an approximately 1:1 ratio of Tyr10 and Tyr13 labeled glucagon. Met27 is in its native thioether form.
List Price : 2067.00 USD
PerkinElmer

SPA Imaging Select-a-Bead Kit, 6 X 500 MG

SPA bead selection kit containing beads for receptor binding studies (contains 500 mg of WGA PS, WGA YOx, WGA PEI type A, WGA PEI type B, PEI PS and poly-L-lysine beads)
List Price : 387.00 USD
List Price : 1903.00 USD
PerkinElmer

Membrane Target Systems: Galanin Gal1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Insulin (porcine), Receptor Grade, [125I]TyrA14], 50µCi

[125I]TyrA14 Insulin has been proven to be active in a receptor binding assay using cultured human fibroblasts as described.8 It may also be used in radioimmunoassay.
List Price : 2143.00 USD
PerkinElmer

Norepinephrine Transporter (human) Cell Line

Our stable recombinant cell lines express a variety of receptors for binding and functional assays.
List Price : 17200.00 USD

Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 1238.00 USD

Hydroxytryptamine Creatinine Sulfate, (Serotonin), 5-[1,2-3H(N)]-, 5-5mCi (185MBq)

5 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.
List Price : 1752.00 USD
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-6 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Serotonin 5HT1a (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from cells stably-transfected with human serotonin 5HT1a receptor
List Price : 891.00 USD
Receptor-expressing cell lines

ValiScreen Leukotriene BLT1 (LTB4R1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

ProfilerPro Kinase Peptide Substrate 5, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 5 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
Receptor-expressing cell lines

ValiScreen Adenosine A3 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-5A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
List Price : 2002.00 USD

Pyrilamine (Mepyramine), [pyridinyl 5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [3H] Mepyramine are available for your research.
List Price : 1497.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1908.00 USD
PerkinElmer

Membrane Target Systems: Prokineticin PKR2 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Prokineticin PKR2 receptor, in HEK-293 cells.
List Price : 891.00 USD

α-Dendrotoxin [125I] 10 µCi

NEX434 [125I]- α-Dendrotoxinsare a class of neurotoxins produced by mamba snakes that block particular subtypes of voltage-gated potassium channels in neurons. Dendrotoxins enhance the release of acetylcholine at neuromuscular junctions.
List Price : 1599.00 USD
PerkinElmer

Membrane Target Systems: TRH (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Calcitonin [Tyr22] (salmon), [125I] 10 µCi

NEX423 [125I]-Calcitonin, [Tyr22] (s) is suitable for the use in radioimmunoassay as well as in the radio-receptor assay.
List Price : 846.00 USD

Norepinephrine, Levo-[7-3H]-, 1mCi (37MBq)

1 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research. This product has a scheduled release date for the third Monday in July.
List Price : 2446.00 USD

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 100µCi (3.7MBq)

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]- will now be made available on a fresh lot schedule. NET876100UC and NET876250UC will be available as a fresh lot once a year on March 15 in 2017.

Vasopressin (Linear), V-1A Antagonist (Phenylacetyl1, 0-Me-D-Tyr2, [125I-Arg6]-),10µCi

NEX310 [125I]-Phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 is useful in receptor studies and autoradiography for the localization and characterization of Vasopressin V1A receptors.
List Price : 918.00 USD
PerkinElmer

Polylysine PS Imaging Bead, 2G

Poly-L-lysine SPA beads enhance the binding of negatively-charged membranes to beads.
List Price : 1561.00 USD
Receptor-expressing cell lines

ValiScreen Vasopressin V1b (rat) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Melanocortin MC5 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Melanocortin MC5 receptor, in HEK-293 cells.
List Price : 891.00 USD
Receptor-expressing cell lines

ValiScreen Vasopressin V2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Neurotensin NTS1(Leu194) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human neurotensin NTS1 (Leu194) receptor, 400 units.
List Price : 866.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 15, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 15 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD

Ifenprodil, [Phenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3H]-Ifenprodil are available for your research.
List Price : 1895.00 USD
PerkinElmer

Membrane Target Systems: Galanin Gal2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 838.00 USD

PDGF [125I] (human) 25 µCi

NEX433 [125I]-PDGF BB homodimer has been shown to work in RIA and receptor studies, using CHO cell line transfected with human PDGF B receptor, and human artery smooth muscle cells.
List Price : 1966.00 USD

MIP-1α (human, recombinant), [125I], 5µCi

NEX298 [125I]-MIP-1α is useful in RIA, receptor studies and crosslinking experiments in the research into immune regulation.
List Price : 700.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.
List Price : 775.00 USD

"Receptor Ligand Binding" 1-50 of 756 Products and Services

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