PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 765 Products and Services

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LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-5A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

DICLOFENAC SODIUM[PHENYLACETIC ACID RING- U-14C]

50 µCi quantities of [Phenylacetic Acid Ring - 14C(U)]-Diclofenac Sodium are available for your research.
List Price : 1952.00 USD

Calcitonin [Tyr22] (salmon), [125I] 10 µCi

NEX423 [125I]-Calcitonin, [Tyr22] (s) is suitable for the use in radioimmunoassay as well as in the radio-receptor assay.
List Price : 846.00 USD
PerkinElmer

Membrane Target Systems: Somatostatin sst4 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Somatostatin sst4 receptor, in HEK-293 cells.
List Price : 891.00 USD
Receptor-expressing cell lines

ValiScreen Neurokinin NK2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

ProfilerPro Kinase Peptide Substrate 30, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 30 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
PerkinElmer

Membrane Target Systems: Bombesin BB1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Bombesin BB1 (human) receptor, in CHO-K1 cells.
List Price : 891.00 USD

Paroxetine, [Phenyl-6`-3H]-, 25µCi (925kBq)

25 µCi quantities of [Phenyl-6'-3H]-Paroxetine are available for your research. This product has a scheduled release date for the third Monday in May and November.
List Price : 564.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 6, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 6 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
PerkinElmer
List Price : 1159.00 USD

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 2067.00 USD
List Price : 1892.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 27, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 27 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
Receptor-expressing cell lines

ValiScreen Neuropeptide Y Y2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Verapamil Hydrochloride, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-Verapamil Hydrochloride are available for your research.
List Price : 592.00 USD

Substance-P (9-Sar, 11-Met(O2)), [2-Prolyl-3,4-3H]-, 50µCi (1.85MBq)

50 µCi quantities of tritiated Substance-P are available for your research.
List Price : 2092.00 USD

Paroxetine, [Phenyl-6`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-6'-3H]-Paroxetine are available for your research. This product has a scheduled release date for the third Monday in May and November.
List Price : 2125.00 USD
Receptor-expressing cell lines

ValiScreen Galanin Gal1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Chemoattractant C5a (human varient) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human chemoattractant C5a (human varient) receptor, 400 units.
List Price : 891.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 29, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 29 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
PerkinElmer

Membrane Target Systems: Bombesin BB3 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Bombesin BB3 (human) receptor, in Balb 3T3 cells.
List Price : 891.00 USD

Epidermal Growth Factor (Murine), [125I]-,50µCi

Epidermal growth factor or EGF is a growth factor that plays an important role in the regulation of cell growth, proliferation, and differentiation by binding to its receptor EGFR.
List Price : 1943.00 USD
List Price : 1685.00 USD

Hydroxytryptamine Creatinine Sulfate (Serotonin), 5-[1,2-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.
List Price : 710.00 USD

WIN 35428, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated WIN 35428 are available for your research.
List Price : 671.00 USD

(-)-CGP-12177, [5,7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 1191.00 USD

QUISQUALIC ACID, [3H]

50 µCi quantities of [3H]-Quisqualic Acid are available for your research. This product has a scheduled release date for the third Monday in September.
List Price : 1615.00 USD
PerkinElmer

Membrane Target Systems: Prolactin Rel Peptide PRRP (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
List Price : 957.00 USD

[125I]Tyr0-Corticotropin Releasing Factor (ovine), 50 µCi

NEX217 Corticotropin-releasing hormone (CRH), originally named corticotropin-releasing factor (CRF), and also called corticoliberin, is a polypeptide hormone and neurotransmitter involved in the stress response.
List Price : 2448.00 USD

Iodo-Melatonin, 2-[125I], 50µCi

NEX236 2-[125I]-iodomelatonin has been used to identify, characterize and localize melatonin binding sites in the brain and peripheral tissues.
List Price : 941.00 USD
PerkinElmer

Membrane Target Systems: GABA B1b (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human GABA B1b receptor, 400 units.
List Price : 891.00 USD
Receptor-expressing cell lines

Chemokine CCR1 ValiScreen Cell Line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Chemokine CX3CR1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

IL-6 (human, recombinant), [125I], 25µCi

NEX269 Interleukin-6 (IL-6) is a protein that in humans is encoded by the IL6 gene. IL-6 is an interleukin that acts as both a pro-inflammatory and anti-inflammatory cytokine. It is secreted by T cells and macrophages to stimulate immune response to trauma, especially burns or other tissue damage leading to inflammation.
List Price : 3924.00 USD

Goat anti-rabbit IgG, [125I], 250µCi (9.25MBq)

Affinity purified goat anti-rabbit IgG is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method1 and is purified by gel filtration chromatography. This method predominantly labels tyrosine residues.
List Price : 893.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 1640.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 26, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 26 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
List Price : 962.00 USD
Price Range : 15300.00 USD - 24400.00 USD
PerkinElmer

Membrane Target Systems: Transporter Serotonin (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Transporter Serotonin receptor, in HEK-293 cells.
List Price : 891.00 USD

WIN 35428, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated WIN 35428 are available for your research.
List Price : 2222.00 USD

AB-MECA, [125I]-(4-Amino-3-[125I]iodobenzyl-5`-N-)-, 10µCi

AB-MECA is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1133.00 USD

"Receptor Ligand Binding" 1-50 of 765 Products and Services

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