PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 763 Products and Services

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MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.
LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.
PerkinElmer

Membrane Target Systems: Serotonin 5HT1a (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from cells stably-transfected with human serotonin 5HT1a receptor
List Price : 891.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 4, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 4 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD

LH-RH, [125I]-[D-Trp6]-, 10µCi

NEX365 [125I]-[D-Trp6]-LH-RH will be useful for receptor binding studies in cell lines and tissue cultures.
List Price : 997.00 USD

QRFP-43, [125I], Human Radioligand, 10µCi (370kBq)

QRFP-43 is a 43 amino acid polypeptide starting from N-terminal pyroglutamic acid and ending at C-terminal arginine-phenylalanine-amide. The intravenous administration of QRFP-43 caused the release of aldosterone, suggesting that QRFP and its receptor have a regulatory function in the rat adrenal gland.
List Price : 1162.00 USD
PerkinElmer

CGP 39653, [Propyl-2,3,3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 1973.00 USD
Receptor-expressing cell lines

ValiScreen KiSS-1 (GPR54) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

α-Bungarotoxin, [125I]-Tyr54-, 250µCi (9.25MBq)

α-bungarotoxin extracted from venom of the Taiwanese banded krait (Bungarus multicinctus) binds the nicotinic acetylcholine receptor found at the neuromuscular junction and the 7 nicotinic acetylcholine receptor in the brain.
List Price : 1232.00 USD
Receptor-expressing cell lines

ValiScreen Vasopressin V1b (rat) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Vasopressin V2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human Vasopressin V2 receptor, 400 units.
List Price : 891.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 14, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 14 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
Receptor-expressing cell lines

ValiScreen N-formyl Peptide (FPRL1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Cholecystokinin Octapeptide, [125I]-, Bolton-Hunter Labeled, 10µCi

NEX203 CCK-8 mediates a number of physiological processes, including digestion and satiety. It is located in the small intestine, and detects the presence of fat in the chyme. As a neuropeptide, CCK mediates satiety by acting on the CCK receptors distributed widely throughout the central nervous system.
List Price : 979.00 USD

2'-deoxycytidine-5'-triphosphate, 5-[125I]Iodo-

Deoxycytidine triphosphate (dCTP) is a nucleoside triphosphate that is used whenever DNA is synthesized, such as in the polymerase chain reaction. 125I dCTP may be used to produce cDNA transcripts of viral or mRNA.
List Price : 1631.00 USD
PerkinElmer

Streptavidin PVT 2G

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 10100.00 USD
PerkinElmer

Membrane Binding YOX Beads, 2G

SPA beads designed for receptor binding studies.
List Price : 463.00 USD

Dihydroalprenolol Hydrochloride, Levo-[Ring, Propyl-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of Levo-[Ring, Propyl-3H(N)]-Dihydroalprenolol Hydrochloride are available for your research.
List Price : 2024.00 USD
PerkinElmer

Membrane Target Systems: Calcitonin CGRP1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
List Price : 957.00 USD
PerkinElmer

Membrane Target Systems: Galanin Gal2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
PerkinElmer

Dopamine Transporter (human) Cell Line

Our stable recombinant cell lines express a variety of receptors for binding and functional assays.
List Price : 17200.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 24, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 24 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
PerkinElmer

Membrane Target Systems: Histamine H2 (human) membrane preparation, in HEK-293 cells. 400 Units.

Cell membranes prepared from HEK293 cells stably transfected with human Histamine H2 receptor, 400 units.
List Price : 891.00 USD
PerkinElmer

ProfilerPro Kinase Peptide Substrate 18, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 18 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 721.00 USD
PerkinElmer

Membrane Target Systems: Vasopressin V1b (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human Vasopressin V1b receptor, 400 units.
List Price : 891.00 USD
Receptor-expressing cell lines

Chemokine CCR1 ValiScreen Cell Line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

WGA PVT PEI TYPE A 500 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.
List Price : 776.00 USD

Peptide YY, (Porcine), ([125I]-PYY), 50µCi

NEX240 Synthetic Peptide YY is radioiodinated with no-carrier-added 125I using a modification of the chloramine-T method.
List Price : 2215.00 USD

MK-912, [3H(G)]

This compound replaces NET1059. MK-912 is an alpha-2 adrenoceptor antagonist. This novel alpha-2 adrenoceptor antagonist radioligand [3H]-MK912 may be used in studies of the regulation of cardiovascular and CNS function.
List Price : 361.00 USD

Somatostatin-14 (human, recombinant), Receptor Grade, 50µCi

NEX446 Tyr11 Somatostatin-14 is radioiodinated with no-carrier-added 125I using amodified lactoperoxidase procedure and is purified by reversed phase HPLC. This method predominantly labels tyrosine residues.
List Price : 2083.00 USD
Receptor-expressing cell lines

ValiScreen Histamine H1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Copper HIS-Tag YSI 125MG

SPA (scintillation proximity assay) beads designed for the capture of His-tagged proteins and peptides.
List Price : 776.00 USD
PerkinElmer

Membrane Target Systems: Serotonin 5HT5a (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Serotonin 5-HT5a receptor, in HEK-293 cells.
List Price : 891.00 USD

Thyroxine, ([125I]-T4), L-[125I]-, 500µCi (18.5MBq), Specific Activity: 135-165µCi (5.00-6.11MBq)/µg

NEX111 L-3,5-Diiodothyronine is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1730.00 USD
PerkinElmer

Membrane Target Systems: Calcitonin AM2 (ADM) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 891.00 USD
PerkinElmer

Membrane Target Systems: Ghrelin (human) membrane preparation, inCHO-K1 cells. 400 Units

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 786.00 USD
PerkinElmer

Protein A PVT 500 MG

Protein A-coated SPA beads, for capturing antibodies in proximity-based radiometric scintillation assays.
List Price : 776.00 USD

CP 55940, [Side Chain-2,3,4-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Side Chain-2, 3, 4-3H(N)]-CP 55940 are available for your research.
List Price : 1823.00 USD

S365057, [Tyr 125I], 10 µCi

NEX396 S36057 is radioiodinated with no carrier added 125I using a lactoperoxidase procedure and is purified by reversed phase HPLC.
List Price : 1249.00 USD
Receptor-expressing cell lines

ValiScreen Somatostatin sst1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

"Receptor Ligand Binding" 1-50 of 763 Products and Services

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