PerkinElmer

Ligands

OF

Eliminate the need for antibodies and reduce assay time with direct detection using our radiolabeled ligands, which provide for sensitive and quantitative measurement of binding.

  • High specific activity — The majority of our 125I-labeled ligands are offered at maximum specific activity. This means virtually every molecule of ligand provided in the stock vial is radiolabeled. For tritiated ligands (3H ligands), pick a ligand with specific activity above 20 Ci/mmol – all of our tritiated ligands meets or exceeds these requirements.
  • High purity — We offer highly-pure radioligands for the highest specific signal with low background in binding assays.
  • High selectivity — Our broad portfolio of agonists and antagonists offers many options for choosing the most selective compound for your receptor.
  • Validated for receptor binding — all of our radioligand products are tested for receptor binding during development. Additionally, many of our radioligands are used to QC our GPCR and receptor cell lines and cell membrane products.

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Application
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Concentration
  • 1 mCi/mL (5)
  • 1.0 - 10 mCi/mL (85)
  • 1.0 - 10 µCi/mL (3)
  • 1.0 mCi/mL (1)
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Detection Method
  • Radiometric (201)
Label Position
  • Generally Labeled (11)
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  • Uniformly Labeled (1)
Product Brand Name
  • NEN Radiochemicals (201)
Radionuclide
  • 14C (9)
  • 33P (1)
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Radioisotope
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  • H-3 (196)
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Volume
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"Ligands" 1-50 of 208 Products and Services

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Cyclopentyl-1,3-Dipropylxanthine, 8-[Dipropyl-2,3-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Cyclopentyl-1, 3-Dipropylxanthine, 8-[Dipropyl-2, 3-3H(N)]- (DPCPX) are available for your research.
List Price : 1238.00 USD

Hydroxytryptamine Creatinine Sulfate, (Serotonin), 5-[1,2-3H(N)]-, 5-5mCi (185MBq)

5 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.
List Price : 1752.00 USD

Pyrilamine (Mepyramine), [pyridinyl 5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [3H] Mepyramine are available for your research.
List Price : 1497.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1908.00 USD

Norepinephrine, Levo-[7-3H]-, 1mCi (37MBq)

1 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research. This product has a scheduled release date for the third Monday in July.
List Price : 2446.00 USD

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 100µCi (3.7MBq)

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]- will now be made available on a fresh lot schedule. NET876100UC and NET876250UC will be available as a fresh lot once a year on March 15 in 2017.

Ifenprodil, [Phenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3H]-Ifenprodil are available for your research.
List Price : 1895.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.
List Price : 775.00 USD

Ro 15-1788, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Ro 15-1788 are available for your research.
List Price : 2045.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 250µCi (9.25MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 3369.00 USD

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 2067.00 USD

Imipramine Hydrochloride, [Benzene ring-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Imipramine hydrochloride are available for your research.
List Price : 1403.00 USD

GBR 12935, [Propylene-2,3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated GBR 12935 are available for your research.
List Price : 2032.00 USD

COUMARIN, 7-ETHOXY, [3- 14C]-

50 µCi quantities of 7-ETHOXY-[3-14C]-Coumarin are available for your research.
List Price : 1850.00 USD

Kainic acid, [Isopropenyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Kainic acid are available for your research.
List Price : 541.00 USD

Colchicine, [ring C, Methoxy-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [ring C, Methoxy-3H]-Colchicine are available for your research.
List Price : 1641.00 USD

WIN 35428, [N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of tritiated WIN 35428 are available for your research.
List Price : 4812.00 USD

Ketanserin Hydrochloride (R41 468), [Ethylene-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Ketanserin hydrochloride are available for your research.
List Price : 585.00 USD

Enkephalin (2-D-Alanine-5-D-Leucine), [Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Enkephalin (2-D-Alanine-5-D-Leucine), [Tyrosyl-3, 5-3H(N)]-, (DADLE) are available for your research.
List Price : 1530.00 USD

Nitrendipine, [5-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Nitrendipine are available for your research.
List Price : 688.00 USD

Prazosin, [7-Methoxy-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [7-Methoxy-3H]-Prazosin are available for your research.
List Price : 2205.00 USD

MK-801, (+)-[3-3H]-%, 25µCi (925kBq)

25 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 618.00 USD

DICLOFENAC SODIUM[PHENYLACETIC ACID RING- U-14C]

50 µCi quantities of [Phenylacetic Acid Ring - 14C(U)]-Diclofenac Sodium are available for your research.
List Price : 1952.00 USD

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 5300.00 USD

SR141716A, [3H]

250 µCi quantities of [3H]-SR141716A are available for your research.
List Price : 2363.00 USD

DOFETILIDE, [N-METHYL-3H], 100 µCi

100 µCi quantities of tritiated Dofetilide are available for your research.
List Price : 1500.00 USD

Deltorphin II(2-D-Ala), [Tyrosyl-3,5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-3, 5-3H]-Deltorphin II (2-D-Ala) are available for your research.
List Price : 3515.00 USD

SCH 23390, [N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.
List Price : 2709.00 USD

Caffeine, [1-Methyl-14C]-, 50µCi (1.85MBq)

50 quantities of [1-Methyl-14C]-Caffeine are available for your research.
List Price : 777.00 USD

SCH 23390, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.
List Price : 1648.00 USD

Spiperone (Spiroperidol), [Benzene ring-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Benzene ring-3H]-Spiperone (Spiroperidol) are available for your research.
List Price : 1559.00 USD

Glibenclamide, Glyburide, [Cyclohexyl-2,3-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Glibenclamide, Glyburide are available for your research.
List Price : 1881.00 USD

Diprenorphine [15,16-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [15, 16-3H]-Diprenorphine are available for your research.
List Price : 953.00 USD

Astemizole, [O-Methyl-3H]-, 25µCi (925kBq)

Astemizole, [O-Methyl-3H]- will now be made available on a fresh lot schedule. NET1140025UC, NET1140250UC, and NET1140001MC will be available as a fresh lot twice a year on March 6 and August 7 in 2017.
List Price : 667.00 USD

Vasopressin (8-L-Arginine), [Phenylalanyl-3,4,5-3H(N)]

250 µCi quantities of [Phenylalanyl-3,4,5-3H(N)]-Vasopressin (8-L-arginine) are available for your research.
List Price : 1822.00 USD

NAAG, [Glutamate-3,4-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [Glutamate-3, 4-3H]-NAAG are available for your research.
List Price : 1035.00 USD

Vinorelbine sulphate, [3H(G)]-

Vinorelbine (trade name Navelbine) is an anti-mitotic chemotherapy drug that is given as a treatment for some types of cancer, including breast cancer and non-small cell lung cancer. Vinorelbine is the first 5´NOR semi-synthetic vinca alkaloid.
List Price : 2517.00 USD

5-HYDROXY TRYPTAMINE, [3H]-

Serotonin (often referred to as 5-HT, short for 5-Hydroxy Tryptamine is a naturally occurring neurotransmitter which is tied to positive mood, certain involuntary muscle control, and countless other functions.
List Price : 1734.00 USD

Dihydroalprenolol Hydrochloride, Levo-[Ring, Propyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[Ring, Propyl-3H(N)]-Dihydroalprenolol Hydrochloride are available for your research.
List Price : 933.00 USD

Enkephalin, [Tyrosyl-2,6-3H(N)]- (2-D-Penicillamine, 5-D-Penicillamine) (DPDPE), 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-2, 6-3H(N)]-Enkephalin (2-D-Penicillamine, 5-D-Penicillamine), (DPDPE) are available for your research.
List Price : 3628.00 USD

TAURINE, [2,2-3H]

1 mCi quantities of tritiated taurine are available for your research.
List Price : 3044.00 USD

Neurotensin, [3,11-Tyrosyl-3,5-3H(N)]-, 25µCi (925kBq)

25 µCi quantities of [3, 11-Tyrosyl-3, 5-3H(N)]-Neurotensin are available for your research.
List Price : 554.00 USD

WAY100635, [METHOXY-3H], 250 uCi

250 µCi quantities of [METHOXY-3H]-WAY100635 are available for your research.
List Price : 2797.00 USD

MELATONIN, [0-METHYL-3H]

250 µCi quantities of [0-METHYL-3H]-MELATONIN are available for your research.
List Price : 2184.00 USD

Pirenzepine, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Pirenzepine are available for your research.
List Price : 1763.00 USD

(+)-Pentazocine, [Ring-1,3-3H]-,250µCi (9.25MBq)

250 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 1926.00 USD

Raclopride, [Methoxy-3H]-, 1mCi (37MBq)

Raclopride, [Methoxy-3H]- will now be made available on a fresh lot schedule. NET975025UC, NET975250UC, and NET975001MC will be available as a fresh lot twice a year on February 6 and August 7 in 2017.
List Price : 4245.00 USD

CGS 21680, [Carboxyethyl-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 4204.00 USD

Norepinephrine, Levo-[ring-2,5,6-3H]-, 5mCi (185MBq)

5 mCi quantities of Levo-[ring-2, 5, 6-3H]-Norepinephrine are available for your research.
List Price : 7300.00 USD

Cytisine HCl, [3,5-3H(N)]-, 250µCi (9.25MBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 2038.00 USD

"Ligands" 1-50 of 208 Products and Services

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