Ligands

OF

Eliminate the need for antibodies and reduce assay time with direct detection using our radiolabeled ligands, which provide for sensitive and quantitative measurement of binding.

  • High specific activity — The majority of our 125I-labeled ligands are offered at maximum specific activity. This means virtually every molecule of ligand provided in the stock vial is radiolabeled. For tritiated ligands (3H ligands), pick a ligand with specific activity above 20 Ci/mmol – all of our tritiated ligands meets or exceeds these requirements.
  • High purity — We offer highly-pure radioligands for the highest specific signal with low background in binding assays.
  • High selectivity — Our broad portfolio of agonists and antagonists offers many options for choosing the most selective compound for your receptor.
  • Validated for receptor binding — all of our radioligand products are tested for receptor binding during development. Additionally, many of our radioligands are used to QC our GPCR and receptor cell lines and cell membrane products.

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"Ligands" 1-50 of 253 Products and Services

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NAAG, [Glutamate-3,4-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [Glutamate-3, 4-3H]-NAAG are available for your research.

List Price: 900.00 USD

Hydroxytryptamine Binoxalate (Serotonin Binoxalate), 5-[2-14C]-, 50µCi (1.85MBq)

50 µCi quantities of 5-[2-14C]-Hydroxytryptamine Binoxalate (Serotonin Binoxalate) are available for your research.

List Price: 631.00 USD

R(+)7-HYDROXY DPAT, [3H], 250 µCi

The standard selective 5-HT1A agonist. Also has moderate affinity for 5-HT7 receptors

List Price: 2489.00 USD

Epinephrine, Levo-[N-methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[N-methyl-3H]-Epinephrine are available for your research.

List Price: 1440.00 USD

Diltiazem, cis-(+)-[N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of cis-(+)-[N-Methyl-3H]-Diltiazem are available for your research.

List Price: 406.00 USD

Hydroxytryptamine Creatinine Sulfate (Serotonin), 5-[1,2-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.

List Price: 618.00 USD

Acetylcholine Iodide, [acetyl-3H], 1mCi (37MBq)

1 mCi quantities of Acetylcholine Iodide, [acetyl-3H]- are available for your research.

List Price: 1199.00 USD

YM-09151-2, [N-Methyl-3H]-, 250mCi (37MBq)

250 µCi quantities of [N-Methyl-3H]-YM-09151-2 are available for your research.

List Price: 1767.00 USD

Ro 15-1788, [N-Methyl-3H]-, 1MC

1 mCi quantities of [N-Methyl-3H]-Ro 15-1788 are available for your research.

List Price: 4023.00 USD

Diltiazem, cis-(+)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of cis-(+)-[N-Methyl-3H]-Diltiazem are available for your research.

List Price: 3043.00 USD

Ro 5-4864, [N-Methyl-3H]-,>97%, 250µCi (9.25MBq)

250 µCi quantities of Ro 5-4864 are available for your research.

List Price: 1597.00 USD

Hydroxytryptamine Binoxalate (Serotonin Binoxalate), 5-[2-14C]-, 250µCi (9.25MBq)

250 µCi quantities of 5-[2-14C]-Hydroxytryptamine Binoxalate (Serotonin Binoxalate) are available for your research.

List Price: 2705.00 USD

SCH 23390, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.

List Price: 1433.00 USD

Paroxetine, [Phenyl-6`-3H]-, 25µCi (925kBq)

25 µCi quantities of [Phenyl-6'-3H]-Paroxetine are available for your research.

List Price: 490.00 USD

U-69,593, [Phenyl-3,4-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3, 4-3H]-U-69,593 are available for your research.

List Price: 1865.00 USD

SCH 23390, [N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.

List Price: 2356.00 USD

MK-912, [3H(G)]

This compound replaces NET1059. MK-912 is an alpha-2 adrenoceptor antagonist. This novel alpha-2 adrenoceptor antagonist radioligand [3H]-MK912 may be used in studies of the regulation of cardiovascular and CNS function.

List Price: 2182.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.

List Price: 2165.00 USD

MDL105,519, [3H]

250 µCi quantities of [3H]-MDL105,519 are available for your research.

List Price: 2178.00 USD

Caffeine, [1-Methyl-14C]-, 50µCi (1.85MBq)

50 quantities of [1-Methyl-14C]-Caffeine are available for your research.

List Price: 676.00 USD

Ro 15-1788, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-Ro 15-1788 are available for your research.

List Price: 537.00 USD

CGP 39653, [Propyl-2,3,3H]-, 1mCi (37MBq)

1 mCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research

List Price: 3954.00 USD

Quinuclidinyl Benzilate, L-[Benzilic-4,4`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of L-[Benzilic-4, 4'-3H]-Quinuclidinyl Benzilate are available for your research.

List Price: 1104.00 USD

Norepinephrine, Levo-[7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.

List Price: 990.00 USD

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Ring, Methylenes-3H(N)]-Histamine Dihydrochloride are available for your research.

List Price: 722.00 USD

Batrachotoxinin A 20-α-Benzoate, [Benzoyl-2,5-3H]-, 100µCi (3.7MBq)

100 µCi quantities of tritiated Batrachotoxinin are available for your research.

List Price: 1698.00 USD

Glibenclamide, Glyburide, [Cyclohexyl-2,3-3H(N)]-, 25µCi (925kBq)

25 µCi quantities of Glibenclamide, Glyburide are available for your research.

List Price: 430.00 USD

3-INDOLYLACETIC ACID, [5-3H(N)]-

Indolylacetic acid, also known as IAA, is a heterocyclic compound that is a phytohormone called auxins. IAA has many different effects, as all auxins do, such as inducing cell elongation and cell division with all subsequent results for plant growth and development.

List Price: 978.00 USD

Dihydroxyphenylethylamine (Dopamine), 3,4-[Ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 3, 4-[Ring-2, 5, 6-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.

List Price: 530.00 USD

PK 11195, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-PK 11195 are available for your research.

List Price: 502.00 USD

Hydroxytryptamine Creatinine Sulfate, (Serotonin), 5-[1,2-3H(N)]-, 5-5mCi (185MBq)

5 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.

List Price: 1523.00 USD

EPOXYCHOLESTEROL, 24(S),25-[26,27-(3H)]-, 100 µCi

100 µCi quantities of tritiated Eposycholesterone are available for your research.

List Price: 2329.00 USD

Methyl-4-Phenylpyridinium Acetate, N-[Methyl-3H]-, MPP (+), 250µCi (9.25MBq)

250 µCi quantities of N-[Methyl-3H]-Methyl-4-Phenylpyridinium Acetate, MPP (+) are available for your research.

List Price: 1129.00 USD

TCP, [Piperdyl-3,4-3H(N)]-

250 µCi quantities of [Piperidyl-3,4-3H(N)]-TCP are available for your research.

List Price: 1579.00 USD

Dihydroalprenolol Hydrochloride, Levo-[Ring, Propyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[Ring, Propyl-3H(N)]-Dihydroalprenolol Hydrochloride are available for your research.

List Price: 811.00 USD

NALOXONE, [N-ALLYL-2,3-3H]-

250 µCi quantities of Naloxone, [N-ALLYL-2,3-3H]- are available for your research.

List Price: 1188.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.

List Price: 674.00 USD

Kainic acid, [Isopropenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Kainic acid are available for your research.

List Price: 1646.00 USD

DAMGO, [Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-3, 5-3H(N)]-DAMGO are available for your research.

List Price: 1360.00 USD

Chloramphenicol, [Ring-3,5-3H]-, 1mCi (37MBq)

1 mCi quantities of [Ring-3, 5-3H]-Chloramphenicol are available for your research.

List Price: 3421.00 USD

Methylhistamine Dihydrochloride, N-α-[methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated methylhistamine dihydrochloride are available for your research.

List Price: 732.00 USD

TAURINE, [2,2-3H]

1 mCi quantities of tritiated taurine are available for your research.

List Price: 2647.00 USD

Ifenprodil, [Phenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3H]-Ifenprodil are available for your research.

List Price: 1648.00 USD

CGS 21680, [Carboxyethyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.

List Price: 1516.00 USD

Cytisine HCl, [3,5-3H(N)]-, 25µCi (925kBq)

25 µCi quantities of [3, 5-3H(N)]-Cytisine HCl are available for your research.

List Price: 493.00 USD

Quinuclidinyl Benzilate, L-[Benzilic-4,4`-3H]-, 25µCi (925kBq)

25 µCi quantities of L-[Benzilic-4, 4'-3H]-Quinuclidinyl Benzilate are available for your research.

List Price: 447.00 USD

MK-801, (+)-[3-3H]-%, 25µCi (925kBq)

25 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.

List Price: 537.00 USD

Norepinephrine, Levo-[ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[ring-2, 5, 6-3H]-Norepinephrine are available for your research.

List Price: 1077.00 USD

ROLIPRAM, [METHYL-3H]

250 µCi quantities of R-(-)-[Methyl-3H]-Rolipram are available for your research.

List Price: 2316.00 USD

8-Hydroxy-DPAT, [Propyl-2,3-ring-1,2,3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Propyl-2, 3-ring-1, 2, 3-3H]-8-Hydroxy-DPAT are available for your research.

List Price: 993.00 USD

"Ligands" 1-50 of 253 Products and Services

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