PerkinElmer

Ligands

OF

Eliminate the need for antibodies and reduce assay time with direct detection using our radiolabeled ligands, which provide for sensitive and quantitative measurement of binding.

  • High specific activity — The majority of our 125I-labeled ligands are offered at maximum specific activity. This means virtually every molecule of ligand provided in the stock vial is radiolabeled. For tritiated ligands (3H ligands), pick a ligand with specific activity above 20 Ci/mmol – all of our tritiated ligands meets or exceeds these requirements.
  • High purity — We offer highly-pure radioligands for the highest specific signal with low background in binding assays.
  • High selectivity — Our broad portfolio of agonists and antagonists offers many options for choosing the most selective compound for your receptor.
  • Validated for receptor binding — all of our radioligand products are tested for receptor binding during development. Additionally, many of our radioligands are used to QC our GPCR and receptor cell lines and cell membrane products.

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  • 1.0 - 10 µCi/mL (3)
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"Ligands" 1-50 of 225 Products and Services

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SCH 23390, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-SCH 23390 are available for your research.
List Price : 1648.00 USD

AF-DX 384, [2,3-Dipropylamino-3H]-, 250µCi (9.25MBq)

250 µCi quantities of AF-DX 384, [2, 3-Dipropylamino-3H]- are available for your research.
List Price : 1853.00 USD

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 1641.00 USD

Norepinephrine, Levo-[7-3H]-, 1mCi (37MBq)

1 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.
List Price : 2446.00 USD

Nociceptin, [Leucyl-3,4,5-3H], 50µCi (1.85MBq)

50 µCi quantities of [Leucyl-3, 4, 5-3H]-Nociceptin are available for your research.
List Price : 3016.00 USD

Norepinephrine, Levo-[7-3H]-, 5mCi (185MBq)

5 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.
List Price : 7600.00 USD

Quinpirole, [N-Propyl-3H]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 1997.00 USD

CCK-8(SULPHATED), [3H]PROPIONY, 50 µCi

50 µCi quantities of [3H]PROPIONY CCK-8(SULPHATED) are available for your research.
List Price : 1413.00 USD

GR 65630, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [N-Methyl-3H]-GR 65630 are available for your research. 
List Price : 535.00 USD

Raclopride, [Methoxy-3H]-, 250µCi (9.25MBq)

Raclopride, [Methoxy-3H]- will now be made available on a fresh lot schedule. NET975025UC, NET975250UC, and NET975001MC will be available as a fresh lot twice a year on February 6 and August 7 in 2017.
List Price : 1767.00 USD

Lysergic Acid Diethylamide, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Lysergic Acid Diethylamide are available for your research.
List Price : 1876.00 USD

Imipramine Hydrochloride, [Benzene ring-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Imipramine hydrochloride are available for your research.
List Price : 1403.00 USD

Kainic acid, [Isopropenyl-3H]-, 1 mCi (37MBq)

1 mCi quantities of tritiated Kainic acid are available for your research.
List Price : 5000.00 USD

CGP 39653, [Propyl-2,3,3H]-, 1mCi (37MBq)

1 mCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 4547.00 USD

GR 65630, [N-Methyl-3H]-, 250µCi (925kBq)

250 µCi quantities of [N-Methyl-3H]-GR 65630 are available for your research. 
List Price : 2399.00 USD

Nicotine, L-(-)-[N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 1547.00 USD

CGS 21680, [Carboxyethyl-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 4204.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 1640.00 USD

GABAPENTIN [3H]

Gabapentin is a GABA analogue. It was originally developed for the treatment of epilepsy, and currently, gabapentin is widely used to relieve pain, especially neuropathic pain.
List Price : 5100.00 USD

Amino-3-Hydroxy-5-Methylisoxazole-4-Propionic Acid (AMPA), DL-α-[5-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of DL-α-[5-Methyl-3H]- Amino-3-Hydroxy-5-Methylisoxazole-4-Propionic Acid (AMPA) are available for your research.
List Price : 540.00 USD

(+)-Pentazocine, [Ring-1,3-3H]-, 1mCi (37MBq)

1 mCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 4616.00 USD

TCP, [Piperdyl-3,4-3H(N)]-

25 µCi quantities of [Piperidyl-3,4-3H(N)]-TCP are available for your research.
List Price : 540.00 USD

COUMARIN, 7-ETHOXY, [3- 14C]-

50 µCi quantities of 7-ETHOXY-[3-14C]-Coumarin are available for your research.
List Price : 1850.00 USD

YM-09151-2, [N-Methyl-3H]-, 250mCi (37MBq)

250 µCi quantities of [N-Methyl-3H]-YM-09151-2 are available for your research.
List Price : 2032.00 USD

Deltorphin II(2-D-Ala), [Tyrosyl-3,5-3H]-, 50µCi (1.85MBq)

50 µCi quantities of [Tyrosyl-3, 5-3H]-Deltorphin II (2-D-Ala) are available for your research.
List Price : 853.00 USD

Kainic acid, [Isopropenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Kainic acid are available for your research.
List Price : 1893.00 USD

Epinephrine, Levo-[N-methyl-3H]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 1657.00 USD

UK-14,304, [Imidazolyl-4,5-3H]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 2352.00 USD

5-Carboxamidotryptamine, [1,2-3H]-, 25uCi

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 551.00 USD

Bradykinin, [2,3-Prolyl-3,4-3H(N)]-, 50µCi (1.85MBq)

50 µCi quantities of [2, 3-Prolyl-3, 4-3H(N)]-Bradykinin are available for your research.
List Price : 1466.00 USD

CGP 39653, [Propyl-2,3,3H]-, 25µCi (925kBq)

25 µCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 555.00 USD

Ifenprodil, [Phenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3H]-Ifenprodil are available for your research.
List Price : 1895.00 USD

Dihydroxyphenylethylamine (Dopamine), 3,4-[Ring-2,5,6-3H]-, 1mCi (37MBq)

1 mCi quantities of 3, 4-[Ring-2, 5, 6-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 1388.00 USD

Sphingosine-1-phosphate, 33P

Sphingosine-1-phosphate is a bioactive lipid and can be used as an endogenous ligand in sphingosine-1-phosphate (S1P) receptor binding assays.
Price Range : 14900.00 USD - 36900.00 USD
PerkinElmer

CGS 21680, [Carboxyethyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 1744.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3850.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1908.00 USD

Methylspiperone, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated methylspiperone are available for your research.
List Price : 1864.00 USD

8-Hydroxy-DPAT, [Propyl-2,3-ring-1,2,3-3H]-, 1mCi (37MBq)

1 mCi quantities of [Propyl-2, 3-ring-1, 2, 3-3H]-8-Hydroxy-DPAT are available for your research.
List Price : 2768.00 USD

AH5183, L-[PIPERIDINYL-3,4-3H]-(VESAMICOL), 250 µCi

Vesamicol (AH5183) an acetylcholine uptake blocker in presynaptic vesicles,reduces the apparent activity of cholinergic neurons, but does not act at the post-synaptic ACh receptor. Vesamicol is a unique tool for investigating presynaptic mechanisms in cholinergic nerve terminals.
List Price : 738.00 USD

WAY100635, [METHOXY-3H], 250 uCi

250 µCi quantities of [METHOXY-3H]-WAY100635 are available for your research.
List Price : 2797.00 USD

Nicotine, L-(-)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 3598.00 USD

(+)-Pentazocine, [Ring-1,3-3H]-, 25µCi (925kBq)

25 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 592.00 USD

PK 11195, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-PK 11195 are available for your research.
List Price : 1905.00 USD

Substance P, [Leucyl-3,4,5-3H(N)]-, 250µCi (9.25MBq)

Note: This product will be discontinued from our catalog portfolio on January 1, 2017.
List Price : 4902.00 USD

Quinuclidinyl Benzilate, L-[Benzilic-4,4`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of L-[Benzilic-4, 4'-3H]-Quinuclidinyl Benzilate are available for your research.
List Price : 1269.00 USD

Diltiazem, cis-(+)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of cis-(+)-[N-Methyl-3H]-Diltiazem are available for your research.
List Price : 3499.00 USD

Neurotensin, [3,11-Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [3, 11-Tyrosyl-3, 5-3H(N)]-Neurotensin are available for your research.
List Price : 2684.00 USD

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 2067.00 USD

Deltorphin II(2-D-Ala), [Tyrosyl-3,5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-3, 5-3H]-Deltorphin II (2-D-Ala) are available for your research.
List Price : 3515.00 USD

"Ligands" 1-50 of 225 Products and Services

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