PerkinElmer

Ligands

OF

Eliminate the need for antibodies and reduce assay time with direct detection using our radiolabeled ligands, which provide for sensitive and quantitative measurement of binding.

  • High specific activity — The majority of our 125I-labeled ligands are offered at maximum specific activity. This means virtually every molecule of ligand provided in the stock vial is radiolabeled. For tritiated ligands (3H ligands), pick a ligand with specific activity above 20 Ci/mmol – all of our tritiated ligands meets or exceeds these requirements.
  • High purity — We offer highly-pure radioligands for the highest specific signal with low background in binding assays.
  • High selectivity — Our broad portfolio of agonists and antagonists offers many options for choosing the most selective compound for your receptor.
  • Validated for receptor binding — all of our radioligand products are tested for receptor binding during development. Additionally, many of our radioligands are used to QC our GPCR and receptor cell lines and cell membrane products.

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Application
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Concentration
  • 1 mCi/mL (5)
  • 1.0 - 10 mCi/mL (85)
  • 1.0 - 10 µCi/mL (3)
  • 1.0 mCi/mL (1)
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Detection Method
  • Radiometric (201)
Label Position
  • Generally Labeled (11)
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Radionuclide
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Radioisotope
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Volume
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"Ligands" 1-50 of 209 Products and Services

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(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 25µCi (925kBq)

25 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research.
List Price : 1640.00 USD

Dihydroxyphenylethylamine [2,5,6,7,8-3H] (Dopamine)

Dopamine receptors have key roles in many processes, including the control of motivation, learning, and fine motor movement, as well as modulation of neuroendocrine signaling.
List Price : 1641.00 USD

(+)-Pentazocine, [Ring-1,3-3H]-,250µCi (9.25MBq)

250 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 1926.00 USD

(-)-CGP-12177, [5,7-3H]-, 25µCi (925kBq)

25 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 488.00 USD

Acetylcholine Iodide, [acetyl-3H], 1mCi (37MBq)

1 mCi quantities of Acetylcholine Iodide, [acetyl-3H]- are available for your research.
List Price : 1318.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3850.00 USD

Cytisine HCl, [3,5-3H(N)]-, 250µCi (9.25MBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 2038.00 USD

Pirenzepine, [N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of [N-Methyl-3H]-Pirenzepine are available for your research.
List Price : 4463.00 USD

(-)-CGP-12177, [5,7-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (-)-CGP-12177, [5,7-3H]- are available for your research.
List Price : 1191.00 USD

Cytisine HCl, [3,5-3H(N)]-, 25µCi (925kBq)

Cytisine HCl, [3,5-3H(N)]- will now be made available on a fresh lot schedule. NET1054025UC and NET1054250UC will be available as a fresh lot once a year on March 6 in 2017.
List Price : 567.00 USD

Ascorbic Acid, L-[1-14C]-,>97%, 50µCi (1.85MBq)

50 µCi quantities of L-[1-14C]-Ascorbic Acid are available for your research.
List Price : 852.00 USD

MELATONIN, [0-METHYL-3H]

250 µCi quantities of [0-METHYL-3H]-MELATONIN are available for your research.
List Price : 2184.00 USD

Retinoic Acid, [11,12-3H]9-cis-

cis-Retinoic Acid may be used in dermatological applications.
List Price : 1997.00 USD

Quinuclidinyl Benzilate, L-[Benzilic-4,4`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of L-[Benzilic-4, 4'-3H]-Quinuclidinyl Benzilate are available for your research.
List Price : 1269.00 USD

3-INDOLYLACETIC ACID, [5-3H(N)]-

Indolylacetic acid, also known as IAA, is a heterocyclic compound that is a phytohormone called auxins. IAA has many different effects, as all auxins do, such as inducing cell elongation and cell division with all subsequent results for plant growth and development.
List Price : 1125.00 USD

COUMARIN, 7-ETHOXY, [3- 14C]-

50 µCi quantities of 7-ETHOXY-[3-14C]-Coumarin are available for your research.
List Price : 1850.00 USD

Norepinephrine, Levo-[ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[ring-2, 5, 6-3H]-Norepinephrine are available for your research.
List Price : 1239.00 USD

TCP, [Piperdyl-3,4-3H(N)]-

250 µCi quantities of [Piperidyl-3,4-3H(N)]-TCP are available for your research.
List Price : 1815.00 USD

QUISQUALIC ACID, [3H]

50 µCi quantities of [3H]-QUISQUALIC ACID are available for your research.
List Price : 1615.00 USD

Thyrotropin Releasing Hormone (3-methyl-histidine2), [L-histidyl-4-3H(N), L-propyl-3,4-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [L-histidyl-4-3H(N), L-propyl-3, 4-3H(N)]-Thyrotropin Releasing Hormone (3-methyl-histidine2) are available for your research.
List Price : 4599.00 USD

Ethylcarboxamidoadenosine, 5`-N-[Adenine-2,8-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 5'-N-[Adenine-2, 8-3H]-Ethylcarboxamidoadenosine (NECA) are available for your research.
List Price : 1477.00 USD

Mazindol, [4`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Mazindol are available for your research.
List Price : 1874.00 USD

17α-HYDROXYPROGESTERONE, [1,2,6,7-3H]

250 µCi quantities of 17a-Hydroxyprogesterone, [1,2,6,7-3H] are available for your research.
List Price : 1136.00 USD

TAURINE, [2,2-3H]

1 mCi quantities of tritiated taurine are available for your research.
List Price : 3044.00 USD

SR 95531, [Butyryl-2,3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Butyryl-2,3-3H]-SR 95531 are available for your research.
List Price : 1765.00 USD

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Ring, Methylenes-3H(N)]-Histamine Dihydrochloride are available for your research.
List Price : 1807.00 USD

Chloramphenicol, [Ring-3,5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Ring-3, 5-3H]-Chloramphenicol are available for your research.
List Price : 1795.00 USD

Deltorphin II(2-D-Ala), [Tyrosyl-3,5-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-3, 5-3H]-Deltorphin II (2-D-Ala) are available for your research.
List Price : 3515.00 USD

Diprenorphine [15,16-3H]-, 25µCi (925kBq)

25 µCi quantities of [15, 16-3H]-Diprenorphine are available for your research.
List Price : 567.00 USD

Raclopride, [Methoxy-3H]-, 250µCi (9.25MBq)

Raclopride, [Methoxy-3H]- will now be made available on a fresh lot schedule. NET975025UC, NET975250UC, and NET975001MC will be available as a fresh lot twice a year on February 6 and August 7 in 2017.
List Price : 1767.00 USD

Astemizole, [O-Methyl-3H]-, 1mCi (37MBq)

Astemizole, [O-Methyl-3H]- will now be made available on a fresh lot schedule. NET1140025UC, NET1140250UC, and NET1140001MC will be available as a fresh lot twice a year on March 6 and August 7 in 2017.
List Price : 6600.00 USD

Pirenzepine, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Pirenzepine are available for your research.
List Price : 1763.00 USD

Substance-P (9-Sar, 11-Met(O2)), [2-Prolyl-3,4-3H]-, 50µCi (1.85MBq)

50 µCi quantities of tritiated Substance-P are available for your research.
List Price : 2092.00 USD

Vinorelbine sulphate, [3H(G)]-

Vinorelbine (trade name Navelbine) is an anti-mitotic chemotherapy drug that is given as a treatment for some types of cancer, including breast cancer and non-small cell lung cancer. Vinorelbine is the first 5´NOR semi-synthetic vinca alkaloid.
List Price : 2517.00 USD

Sphingosine-1-phosphate, 33P

Sphingosine-1-phosphate is a bioactive lipid and can be used as an endogenous ligand in sphingosine-1-phosphate (S1P) receptor binding assays.
Price Range : 14900.00 USD - 36900.00 USD

DTG (1,3-Di-o-tolylguanidine, [p-ring-3H]-), [5-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [5-3H(N)]-DTG (1, 3-Di-o-tolylguanidine, [p-ring-3H]-) are available for your research.
List Price : 5300.00 USD

α-BUNGAROTOXIN,N-[3H]

50 µCi quantities of N-[3H] Alpha-Bungarotoxin are available for your research.
List Price : 3614.00 USD

Thyrotropin Releasing Hormone (3-methyl-histidine2), [L-histidyl-4-3H(N), L-propyl-3,4-3H(N)]-, 50µCi (1.85MBq)

50 µCi quantities of [L-histidyl-4-3H(N), L-propyl-3, 4-3H(N)]-Thyrotropin Releasing Hormone (3-methyl-histidine2) are available for your research.
List Price : 1563.00 USD

Caffeine, [1-Methyl-14C]-, 50µCi (1.85MBq)

50 quantities of [1-Methyl-14C]-Caffeine are available for your research.
List Price : 777.00 USD

(+)-Pentazocine, [Ring-1,3-3H]-, 1mCi (37MBq)

1 mCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 4616.00 USD

SPIPERONE, [3H]

250 µCi quantities of [3H]-Spiperone are available for your research.
List Price : 1718.00 USD

WIN 35428, [N-Methyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated WIN 35428 are available for your research.
List Price : 671.00 USD

Propranolol, L-[4-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated L-propranolol are available for your research.
List Price : 1250.00 USD

Diprenorphine [15,16-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [15, 16-3H]-Diprenorphine are available for your research.
List Price : 953.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.
List Price : 775.00 USD
PerkinElmer

CGS 21680, [Carboxyethyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 1744.00 USD

Hydroxytryptamine Creatinine Sulfate (Serotonin), 5-[1,2-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.
List Price : 710.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 250µCi (9.25MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 3369.00 USD

Norepinephrine, Levo-[7-3H]-, 5mCi (185MBq)

5 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.
List Price : 7600.00 USD

Dihydroxyphenylethylamine, 3,4-[7-3H]-, 1mCi (37MBq)

1 mCi quantities of 3, 4-[7-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 1728.00 USD

"Ligands" 1-50 of 209 Products and Services

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