PerkinElmer

Ligands

OF

Eliminate the need for antibodies and reduce assay time with direct detection using our radiolabeled ligands, which provide for sensitive and quantitative measurement of binding.

  • High specific activity — The majority of our 125I-labeled ligands are offered at maximum specific activity. This means virtually every molecule of ligand provided in the stock vial is radiolabeled. For tritiated ligands (3H ligands), pick a ligand with specific activity above 20 Ci/mmol – all of our tritiated ligands meets or exceeds these requirements.
  • High purity — We offer highly-pure radioligands for the highest specific signal with low background in binding assays.
  • High selectivity — Our broad portfolio of agonists and antagonists offers many options for choosing the most selective compound for your receptor.
  • Validated for receptor binding — all of our radioligand products are tested for receptor binding during development. Additionally, many of our radioligands are used to QC our GPCR and receptor cell lines and cell membrane products.

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Application
  • Drug Discovery & Development (197)
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  • Plant Sciences (1)
Concentration
  • 1 mCi/mL (5)
  • 1.0 - 10 mCi/mL (85)
  • 1.0 - 10 µCi/mL (3)
  • 1.0 mCi/mL (1)
  • <1.0 mCi/mL (10)
Detection Method
  • Radiometric (201)
Label Position
  • Generally Labeled (11)
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  • Uniformly Labeled (1)
Product Brand Name
  • NEN Radiochemicals (202)
Radionuclide
  • 14C (9)
  • 33P (1)
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Radioisotope
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Therapeutic Area
  • Angiogenesis (7)
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"Ligands" 1-50 of 209 Products and Services

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PerkinElmer

CGP 39653, [Propyl-2,3,3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 1973.00 USD

Dihydroalprenolol Hydrochloride, Levo-[Ring, Propyl-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of Levo-[Ring, Propyl-3H(N)]-Dihydroalprenolol Hydrochloride are available for your research.
List Price : 2024.00 USD

MK-912, [3H(G)]

This compound replaces NET1059. MK-912 is an alpha-2 adrenoceptor antagonist. This novel alpha-2 adrenoceptor antagonist radioligand [3H]-MK912 may be used in studies of the regulation of cardiovascular and CNS function.
List Price : 361.00 USD

CP 55940, [Side Chain-2,3,4-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Side Chain-2, 3, 4-3H(N)]-CP 55940 are available for your research.
List Price : 1823.00 USD

Kainic acid, [Isopropenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Kainic acid are available for your research.
List Price : 1893.00 USD

WAY100635, [METHOXY-3H], 250 uCi

250 µCi quantities of [METHOXY-3H]-WAY100635 are available for your research.
List Price : 2797.00 USD

Imipramine Hydrochloride, [Benzene ring-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Imipramine hydrochloride are available for your research.
List Price : 1403.00 USD

Ethylcarboxamidoadenosine, 5`-N-[Adenine-2,8-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 5'-N-[Adenine-2, 8-3H]-Ethylcarboxamidoadenosine (NECA) are available for your research.
List Price : 1477.00 USD

TAURINE, [2,2-3H]

1 mCi quantities of tritiated taurine are available for your research.
List Price : 3044.00 USD

U-69,593, [Phenyl-3,4-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3, 4-3H]-U-69,593 are available for your research.
List Price : 2145.00 USD

AF-DX 384, [2,3-Dipropylamino-3H]-, 250µCi (9.25MBq)

250 µCi quantities of AF-DX 384, [2, 3-Dipropylamino-3H]- are available for your research.
List Price : 1853.00 USD

Cocaine, Levo-[benzoyl-3,4-3H(N)]-

100 µCi and 250 µCi quantities of Levo-[benzoyl-3, 4-3H(N)]-Cocaine are available for your research. 
List Price : 2513.00 USD

Norepinephrine Hydrochloride, DL-[7-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of DL-[7-3H(N)]-Norepinephrine Hydrochloride are available for your research.
List Price : 775.00 USD

Citalopram, [N-Methyl-3H], 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Citalopram are available for your research.
List Price : 2303.00 USD

DAMGO, [Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Tyrosyl-3, 5-3H(N)]-DAMGO are available for your research.
List Price : 1563.00 USD

Methyl-4-Phenylpyridinium Acetate, N-[Methyl-3H]-, MPP (+), 250µCi (9.25MBq)

250 µCi quantities of N-[Methyl-3H]-Methyl-4-Phenylpyridinium Acetate, MPP (+) are available for your research.
List Price : 1299.00 USD

Diltiazem, cis-(+)-[N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of cis-(+)-[N-Methyl-3H]-Diltiazem are available for your research.
List Price : 3499.00 USD

Ascorbic Acid, L-[1-14C]-,>97%, 50µCi (1.85MBq)

50 µCi quantities of L-[1-14C]-Ascorbic Acid are available for your research.
List Price : 852.00 USD

AH5183, L-[PIPERIDINYL-3,4-3H]-(VESAMICOL), 250 µCi

Vesamicol (AH5183) an acetylcholine uptake blocker in presynaptic vesicles,reduces the apparent activity of cholinergic neurons, but does not act at the post-synaptic ACh receptor. Vesamicol is a unique tool for investigating presynaptic mechanisms in cholinergic nerve terminals.
List Price : 738.00 USD

Verapamil Hydrochloride, [N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Verapamil Hydrochloride are available for your research.
List Price : 1978.00 USD

Hemicholinium-3 Diacetate Salt, [Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of  [Methyl-3H]-Hemicholinium-3 Diacetate Salt are available for your research. 
List Price : 2576.00 USD

Rauwolscine, [Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Rauwolscine are available for your research.
List Price : 1628.00 USD

Rosiglitazone, DL- [3H]-

100 µCi quantities of tritiated DL-Rosiglitazone are available for your research.
List Price : 1081.00 USD

Dihydroxyphenylethylamine (Dopamine), 3,4-[Ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of 3, 4-[Ring-2, 5, 6-3H]-Dihydroxyphenylethylamine (Dopamine) are available for your research.
List Price : 609.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 100µCi (3.7MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 1908.00 USD

Iodoantipyrine, 4-[N-Methyl-14C]-, 1mCi (37MBq)

1 mCi quantities of 4-[N-Methyl-14C]-Iodoantipyrine are available for your research.
List Price : 5200.00 USD

PK 11195, [N-Methyl-3H]-, 1mCi (37MBq)

1 mCi quantities of [N-Methyl-3H]-PK 11195 are available for your research.
List Price : 4265.00 USD

Escitalopram, [N-methyl-3H]-

250 µCi quantities of tritiated Escitalopram are available for your research.
List Price : 4063.00 USD

Dihydroalprenolol Hydrochloride, Levo-[Ring, Propyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[Ring, Propyl-3H(N)]-Dihydroalprenolol Hydrochloride are available for your research.
List Price : 933.00 USD

Vasopressin (8-L-Arginine), [Phenylalanyl-3,4,5-3H(N)]

25 µCi quantities of [Phenylalanyl-3,4,5-3H(N)]-Vasopressin (8-L-arginine) are available for your research.
List Price : 600.00 USD

CGS 21680, [Carboxyethyl-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 4204.00 USD

Strychnine, [Benzene-Ring-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Strychnine are available for your research.
List Price : 1882.00 USD

Ifenprodil, [Phenyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-3H]-Ifenprodil are available for your research.
List Price : 1895.00 USD

QUISQUALIC ACID, [3H]

50 µCi quantities of [3H]-Quisqualic Acid are available for your research. This product has a scheduled release date for the third Monday in September.
List Price : 1615.00 USD

Butyl Bicyclophosphorothionate, Tertiary-[35S]-, 250µCi (9.25MBq), Ethanol under nitrogen

35S t-butyl bicyclophosphorothionate (TBPS) is a picrotoxinin analog cage-convulsant that binds GABAA receptors with high affinity and high specificity. Its binding site is closely associated with the chloride ion channel, leading to its classification as a chloride ion channel blocking ligand.
List Price : 3369.00 USD

Norepinephrine, Levo-[ring-2,5,6-3H]-, 250µCi (9.25MBq)

250 µCi quantities of Levo-[ring-2, 5, 6-3H]-Norepinephrine are available for your research.
List Price : 1239.00 USD

NALOXONE, [N-ALLYL-2,3-3H]-

250 µCi quantities of Naloxone, [N-ALLYL-2,3-3H]- are available for your research.
List Price : 1366.00 USD

COUMARIN, 7-ETHOXY, [3- 14C]-

50 µCi quantities of 7-ETHOXY-[3-14C]-Coumarin are available for your research.
List Price : 1850.00 USD

VINBLASTINE SULPHATE, [G-3H]

50 µCi quantities of [G-3H]-Vinblastine Sulphate are available for your research.
List Price : 1430.00 USD

Enkephalin (2-D-Alanine-5-D-Leucine), [Tyrosyl-3,5-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of Enkephalin (2-D-Alanine-5-D-Leucine), [Tyrosyl-3, 5-3H(N)]-, (DADLE) are available for your research.
List Price : 1530.00 USD

Daunomycin, [3H(G)]-, 250µCi (9.25MBq)

250 µCi quantities of [3H(G)]-Daunomycin are available for your research.
List Price : 2390.00 USD

α-BUNGAROTOXIN,N-[3H]

50 µCi quantities of N-[3H] Alpha-Bungarotoxin are available for your research.
List Price : 3614.00 USD

RO 15-4513, [7,9-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated RO 15-4513 are available for your research.
List Price : 2004.00 USD

(+/-)Epibatidine, [5,6-Bicycloheptyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [+/-] [5, 6-Bicycloheptyl-3H]-Epibatidine are available for your research. 
List Price : 3850.00 USD

Iodoantipyrine, 4-[N-Methyl-14C]-, 250µCi (9.25MBq)

250 µCi quantities of 4-[N-Methyl-14C]-Iodoantipyrine are available for your research.
List Price : 2031.00 USD

Kainic acid, [Isopropenyl-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Kainic acid are available for your research.
List Price : 541.00 USD

Methylhistamine Dihydrochloride, N-α-[methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated methylhistamine dihydrochloride are available for your research.
List Price : 841.00 USD

MK-801, (+)-[3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of (+)-[3-3H]-MK-801 are available for your research.
List Price : 2049.00 USD

Nicotine, L-(-)-[N-Methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of L-(-)-[N-Methyl-3H]-Nicotine are available for your research.
List Price : 1547.00 USD

Scopolamine Methyl Chloride, [N-methyl-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [N-Methyl-3H]-Scopolamine Methyl Chloride are available for your research.
List Price : 1440.00 USD

"Ligands" 1-50 of 209 Products and Services

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