| 100-0328 | Binding | Adenosine | A1 (h) |
| 100-0043 | Binding | Adenosine | A2 |
| 100-0003 | Binding | Adenosine | A2A (h) |
| 100-0004 | Binding | Adenosine | A3 |
| 100-0030 | Binding | Adenosine | AD Non selective |
| 300-0214 | Cellular | Adenosine | Transport AOT-T es (h) |
| 300-0215 | Cellular | Adenosine | Transport AOT-T es/cs (h) |
| 100-0047 | Binding | Adenosine | Transporter AOT |
| 100-0001 | Binding | Adenosine | Transporter AOT (h) |
| 100-0106 | Binding | Adenylate Cyclase | Forskolin |
| 300-1118 | Cellular | Adrenergic | Adrenergic, Alpha 2a Agonist (h) |
| 300-1119 | Cellular | Adrenergic | Adrenergic, Alpha 2a Antagonist (h) |
| 100-0100 | Binding | Adrenergic | Alpha 1 Non selective |
| 100-0005 | Binding | Adrenergic | Alpha 1A |
| 100-0006 | Binding | Adrenergic | Alpha 1B |
| 100-0101 | Binding | Adrenergic | Alpha 2 Non selective |
| 100-0007 | Binding | Adrenergic | Alpha 2A (h) |
| 100-0008 | Binding | Adrenergic | Alpha 2B |
| 300-1019 | Cellular | Adrenergic | Alpha 2B, Agonist (h) |
| 300-1020 | Cellular | Adrenergic | Alpha 2B, Antagonist (h) |
| 100-0102 | Binding | Adrenergic | Alpha 2C |
| 100-0009 | Binding | Adrenergic | Alpha 2C (h) |
| 300-0784 | Cellular | Adrenergic | Alpha 2C Agonist (h) |
| 300-0785 | Cellular | Adrenergic | Alpha 2C Antagonist (h) |
| 100-0990 | Binding | Adrenergic | Alpha2b (h) |
| 100-0104 | Binding | Adrenergic | Beta 1 |
| 100-0010 | Binding | Adrenergic | Beta 1 (h) |
| 300-1025 | Cellular | Adrenergic | Beta 1, Agonist (h) |
| 300-1029 | Cellular | Adrenergic | Beta 1, Antagonist (h) |
| 100-0105 | Binding | Adrenergic | Beta 2 |
| 100-0011 | Binding | Adrenergic | Beta 2 (h) |
| 300-0451 | Cellular | Adrenergic | Beta 2 Agonist (h) |
| 300-0452 | Cellular | Adrenergic | Beta 2 Antagonist (h) |
| 100-0325 | Binding | Adrenergic | Beta 3 (h) |
| 100-0103 | Binding | Adrenergic | Beta Non selective |
| 300-0216 | Cellular | Anandamide | Transport AMT-T (h) |
| 100-0084 | Binding | Angiotensin II | AT1 (h) |
| 100-0107 | Binding | Angiotensin II | AT1 Peripheral |
| 300-1056 | Cellular | Angiotensin II | AT1, Agonist (h) |
| 300-1057 | Cellular | Angiotensin II | AT1, Antagonist |
| 100-0108 | Binding | Angiotensin II | AT2 Central |
| 200-0174 | Enzyme | Anhydrase | Isozyme I (h) |
| 200-0175 | Enzyme | Anhydrase | Isozyme II (h) |
| 400-0630 | Cellular | Apoptosis (CASP3) | Blood HL-60 (h) |
| 400-0632 | Cellular | Apoptosis (CASP3) | Blood THP-1 (h) |
| 400-0636 | Cellular | Apoptosis (CASP3) | Brain IMR-32 (h) |
| 400-0643 | Cellular | Apoptosis (CASP3) | Breast MCF7 (h) |
| 400-0644 | Cellular | Apoptosis (CASP3) | Breast T-47D (h) |
| 400-0647 | Cellular | Apoptosis (CASP3) | Colon HT-29 (h) |
| 400-0649 | Cellular | Apoptosis (CASP3) | Lung A549 (h) |
| 400-0656 | Cellular | Apoptosis (CASP3) | Pancreas PANC-1 (h) |
| 400-0658 | Cellular | Apoptosis (CASP3) | Prostate PC-3 (h) |
| 400-0661 | Cellular | Apoptosis (CASP3) | Skin A-431 (h) |
| 100-0109 | Binding | Atrial Naturietic Factor | ANP-A |
| 100-0110 | Binding | Benzodiazepine (peripheral) | Mitochondrial Translocator Protein (TSPO) |
| 100-0111 | Binding | Benzodiazepine (peripheral) | Mitochondrial Translocator Protein (TSPO) (h) |
| 300-0221 | Cellular | Bradykinin | B1 Agonist (h) |
| 300-0283 | Cellular | Bradykinin | B1 Antagonist (h) |
| 100-0012 | Binding | Bradykinin | B2 |
| 300-0222 | Cellular | Bradykinin | B2 Agonist |
| 100-0333 | Binding | Calcium | Type L (a2d Subunit) |
| 100-0113 | Binding | Calcium | Type L (Benzothiazepine Site) |
| 100-0013 | Binding | Calcium | Type L (Dihydropyridine Site) |
| 100-0014 | Binding | Calcium | Type N |
| 100-0073 | Binding | Cannabinoid | CB1 (h) |
| 300-1001 | Cellular | Cannabinoid | CB1, Agonist (h) |
| 300-1002 | Cellular | Cannabinoid | CB1, Antagonist (h) |
| 100-0074 | Binding | Cannabinoid | CB2 (h) |
| 100-0922 | Binding | CAR | Constitutive Androstane Receptor (h) NR1I3 |
| 100-0901 | Binding | CAR | Constitutive Androstane Receptor, Antagonist (h) |
| 300-0551 | Cellular | Cell Surface Marker | CD40, THP1 cells (h) |
| 300-0552 | Cellular | Cell Surface Marker | CD54 (ICAM-1), THP1 cells (h) |
| 300-0553 | Cellular | Cell Surface Marker | CD80 (B7-1), THP1 cells (h) |
| 400-0701 | Cellular | Cellular Anabolism (Protein)td> | Blood HL-60 (h) |
| 400-0707 | Cellular | Cellular Anabolism (Protein) | Brain IMR-32 (h) |
| 400-0714 | Cellular | Cellular Anabolism (Protein) | Breast MCF7 (h) |
| 400-0715 | Cellular | Cellular Anabolism (Protein) | Breast T-47D (h) |
| 400-0717 | Cellular | Cellular Anabolism (Protein) | Colon HCT-116 (h) |
| 400-0718 | Cellular | Cellular Anabolism (Protein) | Colon HT-29 (h) |
| 400-0727 | Cellular | Cellular Anabolism (Protein) | Pancreas PANC-1 (h) |
| 400-0729 | Cellular | Cellular Anabolism (Protein) | Prostate PC-3 (h) |
| 400-0732 | Cellular | Cellular Anabolism (Protein) | Skin A-431 (h) |
| 400-0665 | Cellular | Cellular Metabolism (Glucose) | Blood HL-60 (h) |
| 400-0667 | Cellular | Cellular Metabolism (Glucose) | Blood THP-1 (h) |
| 400-0679 | Cellular | Cellular Metabolism (Glucose) | Breast MCF7 (h) |
| 400-0680 | Cellular | Cellular Metabolism (Glucose) | Breast T-47D (h) |
| 400-0682 | Cellular | Cellular Metabolism (Glucose) | Colon HCT-116 (h) |
| 400-0683 | Cellular | Cellular Metabolism (Glucose) | Colon HT-29 (h) |
| 400-0685 | Cellular | Cellular Metabolism (Glucose) | Lung A549 (h) |
| 400-0692 | Cellular | Cellular Metabolism (Glucose) | Pancreas PANC-1 (h) |
| 400-0694 | Cellular | Cellular Metabolism (Glucose) | Prostate PC-3 (h) |
| 400-0594 | Cellular | Cellular Respiration (ATP/ADP) | Blood HL-60 (h) |
| 400-0596 | Cellular | Cellular Respiration (ATP/ADP) | Blood THP-1 (h) |
| 400-0600 | Cellular | Cellular Respiration (ATP/ADP) | Brain IMR-32 (h) |
| 400-0224 | Cellular | Cellular Respiration (ATP/ADP) | Brain SK-N-MC (h) |
| 400-0578 | Cellular | Cellular Respiration (ATP/ADP) | Breast MCF7 (h) |
| 400-0609 | Cellular | Cellular Respiration (ATP/ADP) | Breast T-47D (h) |
| 400-0611 | Cellular | Cellular Respiration (ATP/ADP) | Colon HCT-116 (h) |
| 400-0612 | Cellular | Cellular Respiration (ATP/ADP) | Colon HT-29 (h) |
| 400-0614 | Cellular | Cellular Respiration (ATP/ADP) | Lung A549 (h) |
| 400-0621 | Cellular | Cellular Respiration (ATP/ADP) | Pancreas PANC-1 (h) |
| 400-0623 | Cellular | Cellular Respiration (ATP/ADP) | Prostate PC-3 (h) |
| 400-0626 | Cellular | Cellular Respiration (ATP/ADP) | Skin A-431 (h) |
| 300-0800 | Cellular | Chemokine | CCR2 Agonist (h) (Ca2+) |
| 300-0801 | Cellular | Chemokine | CCR2 Antagonist (h) (Ca2+) |
| 300-1003 | Cellular | Chemokine | CXCR2, Agonist (h) |
| 300-1004 | Cellular | Chemokine | CXCR2, Antagonist (h) |
| 300-0507 | Cellular | Chemokine | IL-8 (CXCL8) Induction, RPMI cells (h) |
| 300-0499 | Cellular | Chemokine | IL-8 (CXCL8) Induction, THP1 cells (h) |
| 300-0739 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR2/HEK293 cells (h) |
| 300-0741 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR3/HEK293 cells (h) |
| 300-0742 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR4/HEK293 cells (h) |
| 300-0743 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR5/HEK293 cells (h) |
| 300-0744 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR7/HEK293 cells (h) |
| 300-0745 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR8/HEK293 cells (h) |
| 300-0746 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLR9/HEK293 cells (h) |
| 300-0740 | Cellular | Chemokine | IL-8 (CXCL8) Induction, TLRL2/6/HEK293 cells (h) |
| 300-0515 | Cellular | Chemokine | IL-8 (CXCL8) Inhibition, PBMC cells (h) |
| 300-0539 | Cellular | Chemokine | IL-8 (CXCL8) Inhibition, RPMI cells (h) |
| 300-0527 | Cellular | Chemokine | IL-8 (CXCL8) Inhibition, THP1 cells (h) |
| 300-0509 | Cellular | Chemokine | IP-10 (CXCL10) Induction, RPMI cells (h) |
| 300-0500 | Cellular | Chemokine | IP-10 (CXCL10) Induction, THP1 cells (h) |
| 300-0517 | Cellular | Chemokine | IP-10 (CXCL10) Inhibition, PBMC cells (h) |
| 300-0541 | Cellular | Chemokine | IP-10 (CXCL10) Inhibition, RPMI cells (h) |
| 300-0529 | Cellular | Chemokine | IP-10 (CXCL10) Inhibition, THP1 cells (h) |
| 300-0510 | Cellular | Chemokine | MCP-1 (CCL2) Induction, RPMI cells (h) |
| 300-0501 | Cellular | Chemokine | MCP-1 (CCL2) Induction, THP1 cells (h) |
| 300-0518 | Cellular | Chemokine | MCP-1 (CCL2) Inhibition, PBMC cells (h) |
| 300-0542 | Cellular | Chemokine | MCP-1 (CCL2) Inhibition, RPMI cells (h) |
| 300-0530 | Cellular | Chemokine | MCP-1 (CCL2) Inhibition, THP1 cells (h) |
| 300-0511 | Cellular | Chemokine | MIG (CXCL9) Induction, RPMI cells (h) |
| 300-0519 | Cellular | Chemokine | MIG (CXCL9) Inhibition, PBMC cells (h) |
| 300-0543 | Cellular | Chemokine | MIG (CXCL9) Inhibition, RPMI cells (h) |
| 300-0531 | Cellular | Chemokine | MIG (CXCL9) Inhibition, THP1 cells (h) |
| 300-0512 | Cellular | Chemokine | MIP-1a (CCL3) Induction, RPMI cells (h) |
| 300-0503 | Cellular | Chemokine | MIP-1a (CCL3) Induction, THP1 cells (h) |
| 300-0520 | Cellular | Chemokine | MIP-1a (CCL3) Inhibition, PBMC cells (h) |
| 300-0544 | Cellular | Chemokine | MIP-1a (CCL3) Inhibition, RPMI cells (h) |
| 300-0532 | Cellular | Chemokine | MIP-1a (CCL3) Inhibition, THP1 cells (h) |
| 300-0513 | Cellular | Chemokine | MIP-1b (CCL4) Induction, RPMI cells (h) |
| 300-0504 | Cellular | Chemokine | MIP-1b (CCL4) Induction, THP1 cells (h) |
| 300-0521 | Cellular | Chemokine | MIP-1b (CCL4) Inhibition, PBMC cells (h) |
| 300-0545 | Cellular | Chemokine | MIP-1b (CCL4) Inhibition, RPMI cells (h) |
| 300-0533 | Cellular | Chemokine | MIP-1b (CCL4) Inhibition, THP1 cells (h) |
| 300-0514 | Cellular | Chemokine | RANTES (CCL5) Induction, RPMI cells (h) |
| 300-0505 | Cellular | Chemokine | RANTES (CCL5) Induction, THP1 cells (h) |
| 300-0522 | Cellular | Chemokine | RANTES (CCL5) Inhibition, PBMC cells (h) |
| 300-0546 | Cellular | Chemokine | RANTES (CCL5) Inhibition, RPMI cells (h) |
| 300-0534 | Cellular | Chemokine | RANTES (CCL5) Inhibition, THP1 cells (h) |
| 100-0114 | Binding | Cholecystokinin | CCK1 (CCKA) |
| 100-0115 | Binding | Cholecystokinin | CCK2 (CCKB) |
| 300-0217 | Cellular | Choline | Transport CHOL-T |
| 100-0117 | Binding | Complement | Anaphylatoxin C5aR (h) |
| 300-1021 | Cellular | Complement | C5a, Agonist (h) |
| 100-0118 | Binding | Corticotropin Releasing Factor | CRF Non selective |
| 300-0225 | Cellular | Corticotropin Releasing Factor | CRF1 Agonist (h) |
| 300-0293 | Cellular | Corticotropin Releasing Factor | CRF1 Antagonist (h) |
| 400-0905 | Enzyme | CYP19, Aromatase (h) | CYP19, Aromatase (h) |
| 400-0861 | Enzyme | CYP1A1 (h) | CYP1A1 (h) |
| 400-0862 | Enzyme | CYP1A1 (rat) | CYP1A1 (rat) |
| 400-0093 | Enzyme | CYP1A2 (h) | CYP1A2 (h) |
| 400-0864 | Enzyme | CYP1A2 (rat) | CYP1A2 (rat) |
| 400-0863 | Enzyme | CYP1B1 (h) | CYP1B1 (h) |
| 400-0891 | Enzyme | CYP2A1 (rat) | CYP2A1 (rat) |
| 400-0878 | Enzyme | CYP2A2 (rat) | CYP2A2 (rat) |
| 400-0094 | Enzyme | CYP2A6 (h) | CYP2A6 (h) |
| 400-0892 | Enzyme | CYP2B1 (rat) | CYP2B1 (rat) |
| 400-0860 | Enzyme | CYP2B6 (h) | CYP2B6 (h) |
| 400-0882 | Enzyme | CYP2C11 (rat) | CYP2C11 (rat) |
| 400-0885 | Enzyme | CYP2C12 (rat) | CYP2C12 (rat) |
| 400-0883 | Enzyme | CYP2C13 (rat) | CYP2C13 (rat) |
| 400-0868 | Enzyme | CYP2C18 (h) | CYP2C18 (h) |
| 400-0095 | Enzyme | CYP2C19 (h) | CYP2C19 (h) |
| 400-0884 | Enzyme | CYP2C6 (rat) | CYP2C6 (rat) |
| 400-0886 | Enzyme | CYP2C8 (h) | CYP2C8 (h) |
| 400-0096 | Enzyme | CYP2C9*1 (h) | CYP2C9*1 (h) |
| 400-0867 | Enzyme | CYP2D1 (rat) | CYP2D1 (rat) |
| 400-0866 | Enzyme | CYP2D2 (rat) | CYP2D2 (rat) |
| 400-0097 | Enzyme | CYP2D6 (h) | CYP2D6 (h) |
| 400-0876 | Enzyme | CYP2E1 (h) | CYP2E1 (h) |
| 400-0880 | Enzyme | CYP2E1 (rat) | CYP2E1 (rat) |
| 400-0879 | Enzyme | CYP2J2 (h) | CYP2J2 (h) |
| 400-0865 | Enzyme | CYP3A1 (rat) | CYP3A1 (rat) |
| 400-0881 | Enzyme | CYP3A2 (rat) | CYP3A2 (rat) |
| 400-0098 | Enzyme | CYP3A4 (h) | CYP3A4 (h) |
| 400-0869 | Enzyme | CYP3A5 (h) | CYP3A5 (h) |
| 400-0875 | Enzyme | CYP4F12 (h) | CYP4F12 (h) |
| 400-1050 | Enzyme | CYP51 (h) | CYP51 (h) |
| 400-1049 | Enzyme | Cytochrome P450 | Pooled Human Liver Microsome (CYP2C9) |
| 400-0934 | Enzyme | Cytochrome P450 | Pooled Human Liver Microsome (CYP3A4) |
| 300-0794 | Cellular | Cytokine | G-CSF, Induction, PBMC cells (h) |
| 300-0793 | Cellular | Cytokine | GM-CSF Induction, PBMC cells (h) |
| 300-0795 | Cellular | Cytokine | IFNa, Induction, PBMC cells (h) |
| 300-0486 | Cellular | Cytokine | IFNg Induction, PBMC cells (h) |
| 300-0523 | Cellular | Cytokine | IFNg Inhibition, PBMC cells (h) |
| 300-0490 | Cellular | Cytokine | IL-10 Induction, PBMC cells (h) |
| 300-0508 | Cellular | Cytokine | IL-10 Induction, RPMI cells (h) |
| 300-0516 | Cellular | Cytokine | IL-10 Inhibition, PBMC cells (h) |
| 300-0540 | Cellular | Cytokine | IL-10 Inhibition, RPMI cells (h) |
| 300-0791 | Cellular | Cytokine | IL-12p40 Subunit, Induction, THP1 cells (h) |
| 300-0789 | Cellular | Cytokine | IL-12p40 Subunit, Inhibition, THP1 cells (h) |
| 300-0487 | Cellular | Cytokine | IL-1b Induction, PBMC cells (h) |
| 300-0524 | Cellular | Cytokine | IL-1b Inhibition, PBMC cells (h) |
| 300-0488 | Cellular | Cytokine | IL-6 Induction, PBMC cells (h) |
| 300-0498 | Cellular | Cytokine | IL-6 Induction, THP1 cells (h) |
| 300-0525 | Cellular | Cytokine | IL-6 Inhibition, PBMC cells (h) |
| 300-0537 | Cellular | Cytokine | IL-6 Inhibition, THP1 cells (h) |
| 300-0489 | Cellular | Cytokine | IL-8 (CXCL8) Induction, PBMC cells (h) |
| 300-0491 | Cellular | Cytokine | IP-10 (CXCL10) Induction, PBMC cells (h) |
| 300-0492 | Cellular | Cytokine | MCP-1 (CCL2) Induction, PBMC cells (h) |
| 300-0493 | Cellular | Cytokine | MIG (CXCL9) Induction, PBMC cells (h) |
| 300-0502 | Cellular | Cytokine | MIG (CXCL9) Induction, THP1 cells (h) |
| 300-0494 | Cellular | Cytokine | MIP-1a (CCL3) Induction, PBMC cells (h) |
| 300-0495 | Cellular | Cytokine | MIP-1b (CCL4) Induction, PBMC cells (h) |
| 300-0496 | Cellular | Cytokine | RANTES (CCL5) Induction, PBMC cells (h) |
| 300-0497 | Cellular | Cytokine | TNFa Induction, PBMC cells (h) |
| 300-0506 | Cellular | Cytokine | TNFa Induction, THP1 cells (h) |
| 300-0526 | Cellular | Cytokine | TNFa Inhibition, PBMC cells (h) |
| 300-0538 | Cellular | Cytokine | TNFa Inhibition, THP1 cells (h) |
| 200-0921 | Enzyme | Deacetylase | Histone, HDAC3 (h) |
| 200-0925 | Enzyme | Deacetylase | Histone, HDAC6 (h) |
| 200-0956 | Enzyme | Deacetylase | Histone, HDAC8 (h) |
| 200-0926 | Enzyme | Deacetylase | Sirtuin, Sirt1 (h) |
| 200-0927 | Enzyme | Deacetylase | Sirtuin, Sirt2 (h) |
| 200-0928 | Enzyme | Deacetylase | Sirtuin, Sirt3 (h) |
| 200-0997 | Enzyme | Deubiquitinase | BAP1 (h) |
| 200-0994 | Enzyme | Deubiquitinase | UCH-L1 (h) |
| 200-0995 | Enzyme | Deubiquitinase | UCH-L3 (h) |
| 200-0996 | Enzyme | Deubiquitinase | USP5 (h) |
| 100-0120 | Binding | Dopamine | D1 |
| 100-0016 | Binding | Dopamine | D1 (h) |
| 300-0227 | Cellular | Dopamine | D1 Agonist (h) (cAMP) |
| 300-0755 | Cellular | Dopamine | D1 Agonist (h) (Luciferase) |
| 300-0226 | Cellular | Dopamine | D1 Antagonist (h) (Ca2+) |
| 300-0284 | Cellular | Dopamine | D1 Antagonist (h) (cAMP) |
| 300-0757 | Cellular | Dopamine | D1 Antagonist (h) (Luciferase) |
| 100-0121 | Binding | Dopamine | D2 |
| 300-1047 | Cellular | Dopamine | D2L, Agonist (h) |
| 300-1048 | Cellular | Dopamine | D2L, Antagonist (h) |
| 100-1006 | Binding | Dopamine | D2s (h) |
| 100-0018 | Binding | Dopamine | D3 |
| 100-1005 | Binding | Dopamine | D4.2 (h) |
| 100-0019 | Binding | Dopamine | D4.4 (h) |
| 100-0116 | Binding | Dopamine | DA Non-Selective (Clozapine) |
| 300-0331 | Cellular | Dopamine | Transport, DAT-T |
| 100-0015 | Binding | Dopamine | Transporter, DAT |
| 100-0123 | Binding | Dopamine | Transporter, DAT (h) |
| 400-0251 | Cellular | Drug Half-Life | Drug Half-Life |
| 400-0250 | Cellular | Drug Stability | Drug Stability |
| 300-0305 | Cellular | Electron Transfer | Mitochondrial MET |
| 300-0306 | Cellular | Electron Transfer | Reverse Mitochondrial RMET |
| 100-0085 | Binding | Endothelin | ETA (h) |
| 100-0124 | Binding | Endothelin | ETB (h) |
| 100-0125 | Binding | Epidermal Growth Factor | EGF |
| 200-0083 | Enzyme | Esterase | Acetylcholine |
| 200-0327 | Enzyme | Esterase | Acetylcholine (h) |
| 200-0076 | Enzyme | Esterase | Plasma (h) |
| 100-1038 | Binding | Estrogen | Estrogen (bov) |
| 100-1039 | Binding | Estrogen | Estrogen (h) NR3A1 |
| 100-1051 | Binding | Farnesoid | Farnesoid X Receptor (h), Agonist |
| 100-1052 | Binding | Farnesoid | Farnesoid X Receptor (h), Antagonist |
| 100-0023 | Binding | GABA | Chloride TBOB Site |
| 100-0329 | Binding | GABA | GABA Non selective |
| 100-0021 | Binding | GABA | GABA-A Agonist Site |
| 100-0022 | Binding | GABA | GABA-A BDZ Alpha-1 Site |
| 100-1058 | Binding | GABA | GABA-A BDZ Alpha-5 Site |
| 100-0129 | Binding | GABA | GABA-A BDZ Alpha-6 Site |
| 300-0218 | Cellular | GABA | Transport GABA-T |
| 100-0024 | Binding | GABA-B | GABA-B |
| 100-0130 | Binding | Galanin | Galanin Non selective |
| 100-0786 | Binding | GammaHydroxyButyrate | GHB |
| 100-0448 | Binding | Glucocorticoid | Glucocorticoid (h) |
| 100-0026 | Binding | Glutamate | AMPA Site |
| 100-0131 | Binding | Glutamate | Chloride Dependent Site |
| 100-0027 | Binding | Glutamate | Kainate Site |
| 100-0029 | Binding | Glutamate | NMDA Agonist Site |
| 100-0032 | Binding | Glutamate | NMDA Glycine Strychnine-insensitive |
| 100-0028 | Binding | Glutamate | NMDA MK801 Site |
| 100-0031 | Binding | Glutamate | NMDA PCP Site |
| 300-0219 | Cellular | Glutamate | Transport GLUT-T |
| 100-0756 | Binding | Glutamate (metabotropic) | mGluR1 |
| 100-0405 | Binding | Glutamate (metabotropic) | mGluR5 |
| 100-0033 | Binding | Glycine | Glycine Strychnine-sensitive Site |
| 100-0034 | Binding | Histamine | H1 |
| 100-0456 | Binding | Histamine | H1 (h) |
| 300-0998 | Cellular | Histamine | H1, Agonist (h) |
| 300-0999 | Cellular | Histamine | H1, Antagonist (h) |
| 100-0086 | Binding | Histamine | H2 |
| 300-1041 | Cellular | Histamine | H2 Agonist (h) (Ca2+) |
| 300-1040 | Cellular | Histamine | H2 Antagonist (h) (Ca2+) |
| 100-0035 | Binding | Histamine | H3 |
| 300-0229 | Cellular | Histamine | Histamine, H2 Agonist (h) (cAMP) |
| 200-0969 | Enzyme | Hydrolase | FAAH (h) |
| 100-0132 | Binding | Imidazoline | I1 peripheral |
| 100-0075 | Binding | Imidazoline | I2 central |
| 100-0133 | Binding | Inositol Triphosphate | IP3 |
| 200-0924 | Enzyme | Kinase, Lipid | PI3Ka (p110a/p85a) (h) |
| 200-0775 | Enzyme | Kinase, Lipid | Sphingosine SK1 (h) |
| 200-0776 | Enzyme | Kinase, Lipid | Sphingosine SK2 (h) |
| 200-0832 | Enzyme | Kinase, Protein | Abl (E255K) (h) |
| 200-0833 | Enzyme | Kinase, Protein | Abl (G250E) (h) |
| 200-0409 | Enzyme | Kinase, Protein | Abl (h) |
| 200-0834 | Enzyme | Kinase, Protein | Abl (Q252H) (h) |
| 200-0839 | Enzyme | Kinase, Protein | Abl (T315I) (h) |
| 200-0410 | Enzyme | Kinase, Protein | Akt1 (PKBa) (h) |
| 200-0411 | Enzyme | Kinase, Protein | Akt2 (PKBb) (h) |
| 200-0457 | Enzyme | Kinase, Protein | Akt3 (PKBg) (h) |
| 200-0992 | Enzyme | Kinase, Protein | AMPKα1β1γ1(h) |
| 200-0412 | Enzyme | Kinase, Protein | AurA (Aur2/STK6) (h) |
| 200-0812 | Enzyme | Kinase, Protein | AurB (h) |
| 200-0816 | Enzyme | Kinase, Protein | AurC (AURKC) (h) |
| 200-0459 | Enzyme | Kinase, Protein | Axl (h) |
| 200-0920 | Enzyme | Kinase, Protein | BLK (h) |
| 200-0460 | Enzyme | Kinase, Protein | BMX (h) |
| 200-1032 | Enzyme | Kinase, Protein | BRSK1 (h) |
| 200-0769 | Enzyme | Kinase, Protein | BTK (h) |
| 200-0418 | Enzyme | Kinase, Protein | c-Kit (h) |
| 200-0420 | Enzyme | Kinase, Protein | c-TAK (h) |
| 200-0821 | Enzyme | Kinase, Protein | CaMK2a (h) |
| 200-0760 | Enzyme | Kinase, Protein | CaMK2a (rat) |
| 200-0859 | Enzyme | Kinase, Protein | CAMK2d (h) |
| 200-0770 | Enzyme | Kinase, Protein | CaMK4 (h) |
| 200-0989 | Enzyme | Kinase, Protein | CDK1 (h) |
| 200-0414 | Enzyme | Kinase, Protein | CDK2/cyclinA (h) |
| 200-0777 | Enzyme | Kinase, Protein | CDK6 (h) |
| 200-0840 | Enzyme | Kinase, Protein | CDK9/cyclin 1 (h) |
| 200-0480 | Enzyme | Kinase, Protein | CHK1 (CHEK1) (h) |
| 200-0417 | Enzyme | Kinase, Protein | CHK2 (CHEK2) (h) |
| 200-0778 | Enzyme | Kinase, Protein | CK1a (CSNK1A1) (h) |
| 200-0461 | Enzyme | Kinase, Protein | CK1d (CSNK1D) (h) |
| 200-0462 | Enzyme | Kinase, Protein | CK2a1b (h) |
| 200-0774 | Enzyme | Kinase, Protein | cRAF (RAF1) (h) |
| 200-0419 | Enzyme | Kinase, Protein | CSK (h) |
| 200-0815 | Enzyme | Kinase, Protein | DYRK1a (rat) |
| 200-0890 | Enzyme | Kinase, Protein | DYRK1b (h) |
| 200-0422 | Enzyme | Kinase, Protein | DYRK2 (h) |
| 200-0463 | Enzyme | Kinase, Protein | EGFR (ErbB1) (h) |
| 200-1007 | Enzyme | Kinase, Protein | EGFR (L858R) (h) |
| 200-0836 | Enzyme | Kinase, Protein | EGFR (L861Q) (h) |
| 200-0835 | Enzyme | Kinase, Protein | EGFR (T790M) (h) |
| 200-0991 | Enzyme | Kinase, Protein | EGFR (T790M/L858R) (h) |
| 200-1010 | Enzyme | Kinase, Protein | EphA1 (h) |
| 200-0771 | Enzyme | Kinase, Protein | EphA2 (h) |
| 200-0850 | Enzyme | Kinase, Protein | EphA3 (h) |
| 200-0851 | Enzyme | Kinase, Protein | EphA4 (h) |
| 200-0852 | Enzyme | Kinase, Protein | EphA5 (h) |
| 200-0853 | Enzyme | Kinase, Protein | EphA6 (h) |
| 200-0854 | Enzyme | Kinase, Protein | EphA7 (h) |
| 200-0856 | Enzyme | Kinase, Protein | EphA8 (h) |
| 200-0824 | Enzyme | Kinase, Protein | EphB2 (h) |
| 200-0858 | Enzyme | Kinase, Protein | EphB3 (h) |
| 200-0464 | Enzyme | Kinase, Protein | EphB4 (h) |
| 200-0347 | Enzyme | Kinase, Protein | ErbB4 (HER4) (h) |
| 200-0767 | Enzyme | Kinase, Protein | FAK2 (PYK2/PTK2b) (h) |
| 200-1053 | Enzyme | Kinase, Protein | FES (h) |
| 200-0779 | Enzyme | Kinase, Protein | FGFR1 (h) |
| 200-0974 | Enzyme | Kinase, Protein | FGFR3 (h) |
| 200-0802 | Enzyme | Kinase, Protein | FGFR4 (h) |
| 200-0803 | Enzyme | Kinase, Protein | Flt1 (VEGFR1) (h) |
| 200-0831 | Enzyme | Kinase, Protein | Flt3 (D835Y) (h) |
| 200-0423 | Enzyme | Kinase, Protein | Flt3 (h) |
| 200-0804 | Enzyme | Kinase, Protein | Flt4 (VEGFR3) (h) |
| 200-0805 | Enzyme | Kinase, Protein | FMS (CSF1R) (h) |
| 200-0762 | Enzyme | Kinase, Protein | Fyn (h) |
| 200-0424 | Enzyme | Kinase, Protein | GSK-3alpha (h) |
| 200-0425 | Enzyme | Kinase, Protein | GSK-3beta (h) |
| 200-0808 | Enzyme | Kinase, Protein | HGK (ZC1/MAP4K4) (h) |
| 200-0466 | Enzyme | Kinase, Protein | IGF1R (h) |
| 200-0780 | Enzyme | Kinase, Protein | IKKa (h) |
| 200-0772 | Enzyme | Kinase, Protein | IKKb (h) |
| 200-0467 | Enzyme | Kinase, Protein | InsR (h) |
| 200-0972 | Enzyme | Kinase, Protein | InsR (h) - Activation Mode |
| 200-0763 | Enzyme | Kinase, Protein | IRAK4 (h) |
| 200-0465 | Enzyme | Kinase, Protein | Jak2 (h) |
| 200-0933 | Enzyme | Kinase, Protein | Jak3 (h) |
| 200-0773 | Enzyme | Kinase, Protein | JNK2 (h) |
| 200-0768 | Enzyme | Kinase, Protein | KDR (VEGFR2, FLK1) (h) |
| 200-0427 | Enzyme | Kinase, Protein | Lck (h) |
| 200-0842 | Enzyme | Kinase, Protein | LTK (h) |
| 200-0428 | Enzyme | Kinase, Protein | LynA (h) |
| 200-0813 | Enzyme | Kinase, Protein | LynB (h) |
| 200-0747 | Enzyme | Kinase, Protein | MAPK1 (ERK2, p42mapk) (h) |
| 200-0433 | Enzyme | Kinase, Protein | MAPK11 (p38beta) (h) |
| 200-0434 | Enzyme | Kinase, Protein | MAPK12 (p38gamma, SAPK3, ERK6) (h) |
| 200-0435 | Enzyme | Kinase, Protein | MAPK13 (p38delta, SAPK4) (h) |
| 200-0432 | Enzyme | Kinase, Protein | MAPK14 (p38alpha, SAPK2alpha) (h) |
| 200-0754 | Enzyme | Kinase, Protein | MAPK3 (ERK1, p44mapk) (h) |
| 200-0430 | Enzyme | Kinase, Protein | MAPKAPK2 (h) |
| 200-0441 | Enzyme | Kinase, Protein | MAPKAPK5 (PRAK) (h) |
| 200-0826 | Enzyme | Kinase, Protein | MARK1 (h) |
| 200-0987 | Enzyme | Kinase, Protein | MEK1 (MAP2K1) (Human) |
| 200-0983 | Enzyme | Kinase, Protein | MEK2 (MAP2K2) (Human) |
| 200-0855 | Enzyme | Kinase, Protein | MELK (h) |
| 200-0844 | Enzyme | Kinase, Protein | Mer (h) |
| 200-0469 | Enzyme | Kinase, Protein | MET (h) |
| 200-0982 | Enzyme | Kinase, Protein | MKK6, (MAP2K6), (Human) |
| 200-0431 | Enzyme | Kinase, Protein | MSK1 (RPS6KA5) (h) |
| 200-0429 | Enzyme | Kinase, Protein | MST2 (STK3) (h) |
| 200-0918 | Enzyme | Kinase, Protein | MST4 (h) |
| 200-0471 | Enzyme | Kinase, Protein | NEK2 (h) |
| 200-0436 | Enzyme | Kinase, Protein | p70S6K (h) |
| 200-0993 | Enzyme | Kinase, Protein | PAK1 (h) |
| 200-0437 | Enzyme | Kinase, Protein | PAK2 (h) |
| 200-0916 | Enzyme | Kinase, Protein | PAK4 (h) |
| 200-0838 | Enzyme | Kinase, Protein | PDGFa (D842V) (h) |
| 200-0438 | Enzyme | Kinase, Protein | PDGFRa (h) |
| 200-0472 | Enzyme | Kinase, Protein | PDGFRb (h) |
| 200-0439 | Enzyme | Kinase, Protein | PDK1 (h) |
| 200-0906 | Enzyme | Kinase, Protein | Pim1 (h) |
| 200-0473 | Enzyme | Kinase, Protein | Pim2 (h) |
| 200-0440 | Enzyme | Kinase, Protein | PKA (h) |
| 200-0334 | Enzyme | Kinase, Protein | PKC-alpha (h) |
| 200-0335 | Enzyme | Kinase, Protein | PKC-b1 (PRKCB1) (h) |
| 200-0336 | Enzyme | Kinase, Protein | PKC-b2 (PRKCB2) (h) |
| 200-0337 | Enzyme | Kinase, Protein | PKC-d (PRKCD) (h) |
| 200-0346 | Enzyme | Kinase, Protein | PKC-eta (PRKCH) (h) |
| 200-0338 | Enzyme | Kinase, Protein | PKC-g (PRKCG) (h) |
| 200-0807 | Enzyme | Kinase, Protein | PKC-theta (PRKCQ) (h) |
| 200-0765 | Enzyme | Kinase, Protein | PKC-z (PRKCZ) (h) |
| 200-0748 | Enzyme | Kinase, Protein | PKD2 (h) |
| 200-0809 | Enzyme | Kinase, Protein | PKG1a (h) |
| 200-0810 | Enzyme | Kinase, Protein | PKG1b (h) |
| 200-0766 | Enzyme | Kinase, Protein | PLK1 (h) |
| 200-0841 | Enzyme | Kinase, Protein | RET (h) |
| 200-0919 | Enzyme | Kinase, Protein | ROCK1 (h) |
| 200-0442 | Enzyme | Kinase, Protein | ROCK2 (h) |
| 200-0475 | Enzyme | Kinase, Protein | RSK1 (p90RSK/RPS6KA1) (h) |
| 200-0820 | Enzyme | Kinase, Protein | RSK2 (h) |
| 200-0782 | Enzyme | Kinase, Protein | RSK3 (h) |
| 200-0476 | Enzyme | Kinase, Protein | SGK1 (h) |
| 200-0915 | Enzyme | Kinase, Protein | skMLCK (MYLK2) (h) |
| 200-0443 | Enzyme | Kinase, Protein | Src (h) |
| 200-0444 | Enzyme | Kinase, Protein | Syk (h) |
| 200-0827 | Enzyme | Kinase, Protein | Tie2 (h) |
| 200-0783 | Enzyme | Kinase, Protein | TrkA (NTRK1) (h) |
| 200-0811 | Enzyme | Kinase, Protein | TrkB (NTRK2) (h) |
| 200-0819 | Enzyme | Kinase, Protein | TrkC (NTRK3) (h) |
| 200-0814 | Enzyme | Kinase, Protein | TTK (h) |
| 200-0843 | Enzyme | Kinase, Protein | TYRO3 (h) |
| 200-0935 | Enzyme | Kinase, Protein | YES (h) |
| 200-0988 | Enzyme | Kinase, Protein | ZAP70 (h) |
| 100-0036 | Binding | Leukotriene | LTB4 (BLT) |
| 100-0481 | Binding | Leukotriene | LTB4 (BLT1) (h) |
| 100-0482 | Binding | Leukotriene | LTB4 (BLT2) (h) |
| 300-0296 | Cellular | Leukotriene | LTB4 Agonist (h) |
| 300-0297 | Cellular | Leukotriene | LTB4 Antagonist (h) |
| 300-0298 | Cellular | Leukotriene | LTC4/D4 Agonist (h) |
| 100-0037 | Binding | Leukotriene | LTD4 (CysLT1) |
| 300-0749 | Cellular | Lysophospholipid | LPA2 (EDG4) Agonist (h) |
| 300-0750 | Cellular | Lysophospholipid | LPA2 (EDG4) Antagonist (h) |
| 300-0737 | Cellular | Lysophospholipid | Sphingosine-1-phosphate S1P3 (EDG3) Agonist (h) |
| 300-0738 | Cellular | Lysophospholipid | Sphingosine-1-phosphate S1P3 (EDG3) Antagonist (h) |
| 100-0134 | Binding | Melatonin | Melatonin Non selective |
| 100-0893 | Binding | Mineralocorticoid | Mineralocorticoid (rat) |
| 100-0135 | Binding | Muscarinic | M Non selective Central |
| 100-0136 | Binding | Muscarinic | M Non selective Peripheral |
| 100-0137 | Binding | Muscarinic | M1 |
| 100-0038 | Binding | Muscarinic | M1 (h) |
| 300-0231 | Cellular | Muscarinic | M1 Agonist (h) (Ca2+) |
| 300-0454 | Cellular | Muscarinic | M1 Antagonist (h) (Ca2+) |
| 100-0138 | Binding | Muscarinic | M2 |
| 100-0039 | Binding | Muscarinic | M2 (h) |
| 100-0139 | Binding | Muscarinic | M3 |
| 100-0040 | Binding | Muscarinic | M3 (h) |
| 300-0455 | Cellular | Muscarinic | M3 Agonist (h) (Ca2+) |
| 100-0041 | Binding | Muscarinic | M4 (h) |
| 100-0042 | Binding | Muscarinic | M5 (h) |
| 100-0044 | Binding | Neurokinin | NK1 |
| 100-0140 | Binding | Neurokinin | NK2 (NKA) (h) |
| 300-1022 | Cellular | Neurokinin | NK2, Agonist (h) (Ca2+) |
| 300-1000 | Cellular | Neurokinin | NK2, Agonist (h) (LF) |
| 300-1023 | Cellular | Neurokinin | NK2, Antagonist (h) |
| 100-0141 | Binding | Neurokinin | NK3 (NKB) |
| 100-0142 | Binding | Neuropeptide Y | NPY Non selective |
| 100-0143 | Binding | Neuropeptide Y | NPY1 (h) |
| 100-0045 | Binding | Neuropeptide Y | NPY2 (h) |
| 100-0144 | Binding | Neurotensin | NT |
| 100-0145 | Binding | Neurotensin | NT (h) |
| 100-0046 | Binding | Nicotinic | a-BnTx Insensitive Neuronal |
| 100-0359 | Binding | Nicotinic | a-BnTx Insensitive Neuronal (h) |
| 100-0403 | Binding | Nicotinic | a-BnTx Sensitive Muscle-Type (h) |
| 300-0564 | Cellular | Nicotinic | NAG Neuronal Agonist (h) |
| 300-0565 | Cellular | Nicotinic | NAG Neuronal Antagonist (h) |
| 100-0971 | Binding | Nicotinic | α-Bungarotoxin Sensitive, Neuronal (α7) |
| 100-0089 | Binding | Nitric Oxide | NOS (neuronal-binding) |
| 300-0332 | Cellular | Norepinephrine | Transport NET-T |
| 300-0404 | Cellular | Norepinephrine | Transport NET-T (h) |
| 100-0048 | Binding | Norepinephrine | Transporter NET |
| 100-0146 | Binding | Norepinephrine | Transporter NET (h) |
| 100-0149 | Binding | Opioid | Delta |
| 100-0049 | Binding | Opioid | Delta (DOP,OP1) (h) |
| 100-0150 | Binding | Opioid | Kappa 1 |
| 100-0151 | Binding | Opioid | Mu |
| 100-0051 | Binding | Opioid | Mu (h) |
| 300-0234 | Cellular | Opioid | Mu Agonist (h) (GTPgS) |
| 300-0294 | Cellular | Opioid | Mu Antagonist (h) (GTPgS) |
| 100-0072 | Binding | Opioid | Nociceptin, ORL1 (h) |
| 100-0888 | Binding | Opioid | Nociceptin, ORL1 brain (h) |
| 100-0889 | Binding | Opioid | Nociceptin, ORL1 brain (macaque) |
| 100-1024 | Binding | Opioid | Nociceptin, ORL1 brain (Rabbit) |
| 100-0887 | Binding | Opioid | Nociceptin, ORL1 brain (rat) |
| 300-1045 | Cellular | Opioid | Nociceptin, ORL1, Agonist (h) |
| 300-1046 | Cellular | Opioid | Nociceptin, ORL1, Antagonist (h) |
| 100-0147 | Binding | Opioid | OP Non-selective |
| 100-0148 | Binding | Opioid | OP Non-selective (+Na+) |
| 200-0326 | Enzyme | Other | Catechol-O'-Methyl Transferase COMT |
| 200-0176 | Enzyme | Other | Choline Acetyl Transferase ChAT |
| 200-0180 | Enzyme | Other | Glutamic Acid Decarboxylase GAD |
| 300-0792 | Cellular | Other | PGE2, Induction, PBMC cells (h) |
| 300-0790 | Cellular | Other | PGE2, Inhibition, PBMC cells (h) |
| 200-1061 | Enzyme | Oxidase | MAO-A central |
| 200-1060 | Enzyme | Oxidase | MAO-A peripheral |
| 200-0186 | Enzyme | Oxidase | MAO-B central |
| 200-0079 | Enzyme | Oxidase | MAO-B peripheral |
| 200-0177 | Enzyme | Oxygenase | Cyclooxygenase, COX-1 |
| 200-0178 | Enzyme | Oxygenase | Cyclooxygenase, COX-2 |
| 100-0152 | Binding | Oxytocin | Oxytocin |
| 100-0806 | Binding | P-Glyocoprotein (PGP) | Transporter P-Glycoprotein (PGP) (h) |
| 200-1068 | Enzyme | PDE10A1 (h) | PDE10A1 (h) |
| 200-0943 | Enzyme | PDE10A2 (h) | PDE10A2 (h) |
| 200-0954 | Enzyme | PDE11A (h) | PDE11A (h) |
| 200-0966 | Enzyme | PDE1A1 (h) | PDE1A1 (h) |
| 200-1030 | Enzyme | PDE1B (h) | PDE1B (h) |
| 200-1120 | Enzyme | PDE1C (h) | PDE1C (h) |
| 200-0967 | Enzyme | PDE2A (h) | PDE2A1 (h) |
| 200-0962 | Enzyme | PDE3A (h) | PDE3A (h) |
| 200-1031 | Enzyme | PDE3B (h) | PDE3B (h) |
| 200-0941 | Enzyme | PDE4A1A (h) | PDE4A1A (h) |
| 200-0963 | Enzyme | PDE4B1 (h) | PDE4B1 (h) |
| 200-1062 | Enzyme | PDE4C1 (h) | PDE4C1 (h) |
| 200-0986 | Enzyme | PDE4D3 (h) | PDE4D3 (h) |
| 200-1064 | Enzyme | PDE4D7 (h) | PDE4D7 (h) |
| 200-0942 | Enzyme | PDE5A1 (h) | PDE5A1 (h) |
| 200-0968 | Enzyme | PDE7A (h) | PDE7A (h) |
| 200-1066 | Enzyme | PDE7B (h) | PDE7B (h) |
| 200-0958 | Enzyme | PDE8A1 (h) | PDE8A1 (h) |
| 200-0955 | Enzyme | PDE9A2 (h) | PDE9A2 (h) |
| 400-0936 | Solubility | Permeability | Aqueous Compound Solubility |
| 200-0788 | Enzyme | Phosphatase | LMPTP-A (h) |
| 200-0787 | Enzyme | Phosphatase | PP1a (h) |
| 200-0188 | Enzyme | Phosphatase | PP2A (h) |
| 200-0189 | Enzyme | Phosphatase | PP2B (calcineruin) |
| 200-0965 | Enzyme | Phosphatase | PP2Ca (h) |
| 200-0930 | Enzyme | Phosphatase | PTEN (h) |
| 200-0845 | Enzyme | Phosphatase | PTP-BAS (h) |
| 200-0190 | Enzyme | Phosphatase | PTP-CD45 (h) |
| 200-0846 | Enzyme | Phosphatase | PTP-D2 (h) |
| 200-0191 | Enzyme | Phosphatase | PTP-LAR (h) |
| 200-0796 | Enzyme | Phosphatase | PTP-MEG1 (h) |
| 200-0797 | Enzyme | Phosphatase | PTP-MEG2 (h) |
| 200-0870 | Enzyme | Phosphatase | PTP-MU (h) |
| 200-0799 | Enzyme | Phosphatase | PTP-PEST/N12 (h) |
| 200-0798 | Enzyme | Phosphatase | PTP-SHP1 (h) |
| 200-0847 | Enzyme | Phosphatase | PTP-SHP2 (h) |
| 200-0192 | Enzyme | Phosphatase | PTP-T-Cell (h) |
| 200-0092 | Enzyme | Phosphatase | PTP1b (h) |
| 200-0080 | Enzyme | Phosphatase | PTPb (h) |
| 200-0929 | Enzyme | Phosphatase | SHIP2 (h) |
| 200-0193 | Enzyme | Phosphatase | VHR (Dual) (h) |
| 200-1035 | Enzyme | Phosphodiesterases (PDEs) | PDE6C (h) |
| 100-0153 | Binding | Platelet Activating Factor | PAF |
| 300-0236 | Cellular | Platelet Activating Factor | PAF Agonist (h) |
| 100-0052 | Binding | Potassium | ATP Sensitive (KATP) |
| 100-0054 | Binding | Potassium | Ca2+ Activated (VI) |
| 100-0330 | Binding | Potassium | hERG (I[Kr]) (h) |
| 300-0399 | Cellular | Potassium | hERG I[Kr] [Rb+] (h) |
| 100-0914 | Binding | PPAR | Peroxisome Proliferator Activated Receptor, Gamma (h) |
| 100-0873 | Binding | PPAR | Peroxisome Proliferator Activator Alpha (h) |
| 100-0899 | Binding | Pregnane | Pregnane X Receptor, PXR (h) |
| 100-0154 | Binding | Progesterone | Progesterone (bov) |
| 100-0155 | Binding | Progesterone | Progesterone (h) |
| 400-0288 | Cellular | Proliferation | Blood HL-60 (h) |
| 400-0291 | Cellular | Proliferation | Blood THP-1 (h) |
| 400-0308 | Cellular | Proliferation | Brain IMR-32 (h) |
| 400-0247 | Cellular | Proliferation | Breast MCF7 (h) |
| 400-0315 | Cellular | Proliferation | Breast T-47D (h) |
| 400-0318 | Cellular | Proliferation | Colon HCT-116 (h) |
| 400-0289 | Cellular | Proliferation | Colon HT-29 (h) |
| 400-0287 | Cellular | Proliferation | Lung A549 (h) |
| 400-0319 | Cellular | Proliferation | Lung DMS 53 (h) |
| 400-0321 | Cellular | Proliferation | Lung IMR-90 (h) |
| 400-0290 | Cellular | Proliferation | Pancreas PANC-1 (h) |
| 400-0557 | Cellular | Proliferation | Prostate PC-3 (h) |
| 400-0324 | Cellular | Proliferation | Skin A-431 (h) |
| 300-0981 | Cellular | Prostanoid | Prostaglandin E2 (PGE2) Antagonist (h) |
| 300-0980 | Cellular | Prostanoid | Prostaglandin E2 (PGE2) Agonist (h) |
| 200-0931 | Enzyme | Protease | ACE1 (h) |
| 200-0959 | Enzyme | Protease | ADAM10 (h) |
| 200-0407 | Enzyme | Protease | Beta Secretase (h) |
| 200-0196 | Enzyme | Protease | Caspase-1 (h) |
| 200-0203 | Enzyme | Protease | Caspase-10 (h) |
| 200-0081 | Enzyme | Protease | Caspase-2 (h) |
| 200-0082 | Enzyme | Protease | Caspase-3 (h) |
| 200-0197 | Enzyme | Protease | Caspase-4 (h) |
| 200-0198 | Enzyme | Protease | Caspase-5 (h) |
| 200-0201 | Enzyme | Protease | Caspase-8 (h) |
| 200-0202 | Enzyme | Protease | Caspase-9 (h) |
| 200-0204 | Enzyme | Protease | Elastase (h) |
| 200-0909 | Enzyme | Protease | Endothelin Converting Enzyme (ECE1) (h) |
| 200-0910 | Enzyme | Protease | Endothelin Converting Enzyme (ECE2) (h) |
| 200-0205 | Enzyme | Protease | Matrix-Metallo MMP-1 (h) |
| 200-0970 | Enzyme | Protease | Matrix-Metallo MMP-12 (h) |
| 200-0213 | Enzyme | Protease | Matrix-Metallo MMP-13 (h) |
| 200-0206 | Enzyme | Protease | Matrix-Metallo MMP-2 (h) |
| 200-0207 | Enzyme | Protease | Matrix-Metallo MMP-3 (h) |
| 200-0208 | Enzyme | Protease | Matrix-Metallo MMP-7 (h) |
| 200-0210 | Enzyme | Protease | Matrix-Metallo MMP-9 (h) |
| 200-0961 | Enzyme | Protease | Neprilysin (h) |
| 200-0960 | Enzyme | Protease | UPA (h) |
| 100-0156 | Binding | Protein Kinase C | PDBu |
| 100-0157 | Binding | Purinergic | P2Y |
| 100-0055 | Binding | Purinergic | P2Y (h) |
| 300-0238 | Cellular | Purinergic | P2Y2 Agonist (h) |
| 300-0286 | Cellular | Purinergic | P2Y2 Antagonist (h) |
| 100-0923 | Binding | Retinoic Acid | RARa, Agonist (h) |
| 100-0907 | Binding | Retinoic Acid | RARa, Antagonist (h) |
| 100-0877 | Binding | Retinoic Acid | Retinoic Acid Receptor (h) Antagonist Binding |
| 100-0913 | Binding | Retinoic Acid | Retinoic Acid Receptor (rat) |
| 100-0158 | Binding | Serotonin | 5HT Non selective |
| 100-0159 | Binding | Serotonin | 5HT1 Non selective |
| 100-0160 | Binding | Serotonin | 5HT1A |
| 100-0057 | Binding | Serotonin | 5HT1A (h) |
| 300-1011 | Cellular | Serotonin | 5HT1A, Agonist (h) |
| 300-1012 | Cellular | Serotonin | 5HT1A, Antagonist (h) |
| 100-0161 | Binding | Serotonin | 5HT1B |
| 100-0058 | Binding | Serotonin | 5HT1D |
| 100-0162 | Binding | Serotonin | 5HT1D (h) |
| 100-0059 | Binding | Serotonin | 5HT2A |
| 100-0163 | Binding | Serotonin | 5HT2A (h) |
| 300-1054 | Cellular | Serotonin | 5HT2A, Agonist (h) |
| 300-1055 | Cellular | Serotonin | 5HT2A, Antagonist (h) |
| 100-0848 | Binding | Serotonin | 5HT2B (h) |
| 300-1013 | Cellular | Serotonin | 5HT2B Agonist (h) |
| 300-1014 | Cellular | Serotonin | 5HT2B Antagonist (h) |
| 100-0060 | Binding | Serotonin | 5HT2C |
| 300-1008 | Cellular | Serotonin | 5HT2C Agonist (h) |
| 300-1009 | Cellular | Serotonin | 5HT2C Antagonist (h) |
| 100-0061 | Binding | Serotonin | 5HT3 |
| 100-0406 | Binding | Serotonin | 5HT3 (h) |
| 300-0303 | Cellular | Serotonin | 5HT3 Agonist |
| 300-0304 | Cellular | Serotonin | 5HT3 Antagonist |
| 100-0062 | Binding | Serotonin | 5HT4 |
| 100-0063 | Binding | Serotonin | 5HT5A (h) |
| 100-0064 | Binding | Serotonin | 5HT6 (h) |
| 100-0065 | Binding | Serotonin | 5HT7 (h) |
| 300-0220 | Cellular | Serotonin | Transport SERT-T (h) |
| 100-0056 | Binding | Serotonin | Transporter SERT |
| 100-0099 | Binding | Serotonin | Transporter SERT (h) |
| 100-0164 | Binding | Sigma | S Non selective |
| 100-0066 | Binding | Sigma | S1 |
| 100-0067 | Binding | Sigma | S2 |
| 100-0069 | Binding | Sodium | Site 2 |
| 100-0165 | Binding | Somatostatin | SOM Non selective |
| 100-0167 | Binding | Testosterone (Androgen) | Testosterone Cytosolic (h) |
| 100-0168 | Binding | Testosterone (Androgen) | Testosterone Nuclear |
| 100-0070 | Binding | Thromboxane | TXA2 (h) |
| 100-0169 | Binding | Thyrotropin Releasing Hormone | TRH |
| 100-0170 | Binding | Vasoactive Intestinal Peptide | VIP Non selective |
| 100-0171 | Binding | Vasopressin | V1 |
| 100-0172 | Binding | Vasopressin | V1A (h) |
| 100-1028 | Binding | Vasopressin | V2 (h) |
| 300-1015 | Cellular | Vasopressin | V2, Agonist (h) |
| 300-1016 | Cellular | Vasopressin | V2, Antagonist (h) |
| 300-0554 | Cellular | Vesicular Monoamine | Transport VMAT1 |
| 300-0555 | Cellular | Vesicular Monoamine | Transport VMAT2 |
| 100-0751 | Binding | Vesicular Monoamine | Transporter VMAT2 |
| 400-0563 | Cellular | Viability (Live/Dead) | Blood HL-60 (h) |
| 400-0567 | Cellular | Viability (Live/Dead) | Blood THP-1 (h) |
| 400-0571 | Cellular | Viability (Live/Dead) | Brain IMR-32 (h) |
| 400-0578 | Cellular | Viability (Live/Dead) | Breast MCF7 (h) |
| 400-0579 | Cellular | Viability (Live/Dead) | Breast T-47D (h) |
| 400-0340 | Cellular | Viability (Live/Dead) | Colon HCT-116 (h) |
| 400-0341 | Cellular | Viability (Live/Dead) | Colon HT-29 (h) |
| 400-0581 | Cellular | Viability (Live/Dead) | Lung A549 (h) |
| 400-0590 | Cellular | Viability (Live/Dead) | Prostate PC-3 (h) |
| 400-0592 | Cellular | Viability (Live/Dead) | Skin A-431 (h) |