| 5-Hydroxytryptamine |
5-HT1A |
ES-310-C
MCL-508 |
ES-310-A |
|
|
6110501400UA (CHO-K1)
RBHS1AM400UA (HEK293) |
| 5-HT2A |
ES-313-C |
|
ES-313-A |
|
ES-313-M400UA |
| 5-HT2B |
ES-314-C |
|
ES-314-A |
|
ES-314-M400UA |
| 5-HT2C (non edited isoform) |
ES-318-C |
|
ES-318-A |
|
6110548400UA (HEK293) ES-318-M400UA (1321N1) |
| 5-HT2C (edited isoform) |
ES-315-C |
|
ES-315-A |
|
ES-315-M400UA |
| 5-HT5A |
ES-401-C (CHO-K1)
MCL-509 (HEK293) |
|
ES-401-A |
|
RBHS5AM400UA (HEK293) ES-401-M400UA (CHO-K1) |
| 5-HT6 |
ES-316-C |
ES-316-CF |
ES-316-A |
ES-316-AF |
ES-316-M400UA (human) RBHS6M400UA (human) RBRS6M400UA (rat) |
| 5-HT7 |
|
|
|
|
6110512400UA (human) RBRS7M400UA (rat) |
| Acetylcholine (Muscarinic) |
M1 |
ES-210-C |
|
ES-210-A |
ES-210-AF |
RBHM1M400UA |
| M2 |
ES-211-C |
|
ES-211-A |
ES-211-AF |
RBHM2M400UA |
| M3 |
ES-212-C |
|
ES-212-A |
ES-212-AF |
RBHM3M400UA |
| M4 |
ES-213-C |
|
ES-213-A |
ES-213-AF |
RBHM4M400UA |
| M5 |
ES-214-C |
|
ES-214-A |
ES-214-AF |
RBHM5M400UA |
| Adenosin |
A1 |
ES-010-C |
ES-010-CF |
ES-010-A |
ES-010-AF |
ES-010-M400UA (human) 6110511400UA (rat) 6110120400UA (rat) |
| A2A |
ES-011-C
MCL-511 (rat) |
ES-011-CF |
ES-011-A |
|
RBHA2AM400UA |
| A2B |
ES-013-C
RBHA2BC |
ES-013-CF |
ES-013-A |
|
ES-013-M400UA |
| A3 |
ES-012-C MCL-512 (rat) |
|
ES-012-A AX-001-PCF |
ES-012-AF |
ES-012-M400UA RBRA3M400UA |
| Adrenoreceptors |
α1A |
ES-036-C |
|
ES-036-A |
ES-036-AF |
ES-036-M400UA |
| α1B |
|
|
ES-037-A |
|
|
| α1D |
|
|
ES-038-A |
|
|
| α2A |
ES-030-C |
ES-030-CF |
ES-030-A |
ES-030-AF |
ES-033-M400UA (CHO-K1) 6110110400UA (SF9) |
| α2B |
ES-031-C |
|
ES-031-A |
|
ES-031-M400UA |
| α2C |
ES-032-C |
ES-032-CF |
ES-032-A |
|
ES-032-M400UA (CHO-K1) 6110114400UA (SF9) |
| β1 |
ES-033-C |
ES-033-CF |
ES-033-A |
ES-033-AF |
ES-033-M400UA (CHO-K1) 6110110400UA (SF9) |
| β2 |
ES-034-C RBHBE2C |
ES-034-CF |
|
|
ES-034-M400UA (CHO-K1) 6110106400UA (SF9) RBHBE2M400UA (HEK293) |
| β3 |
ES-035-C |
ES-035-CF |
|
|
ES-035-M400UA (CHO-K1) RBHBE3M400UA (SK-N-MC) |
| Anaphylatoxin |
C3a |
ES-730-C |
ES-730-CF |
ES-730-A |
|
ES-730-M400UA |
| C5a |
ES-731-C |
ES-731-CF |
ES-731-A |
ES-731-AF |
ES-731-M400UA 6110526400UA |
| Angiotensin |
AT1 |
ES-072-C |
|
ES-072-A |
ES-072-AF |
ES-072-M400UA 6110121400UA |
| AT2 |
ES-070-C (human) ES-071-C (mouse) |
|
|
|
ES-070-M400UA (human) ES-071-M400UA (mouse) |
| Apelin |
APJ |
ES-460-C |
ES-460-CF |
ES-460-A |
|
ES-460-M400UA |
| Beta Alanine |
MRDPRD, TGR7 |
|
|
ES-741-A |
|
|
| Bombesin |
BB1 |
|
|
ES-581-A |
|
RBHBS1M400UA |
| BB2 |
ES-582-C |
|
ES-582-A |
|
ES-582-M400UA (CHO-K1) RBHBS2M400UA (HEK293) |
| BB3 |
|
|
ES-580-A |
|
RBHBS3M400UA |
| Bradykinin |
B1 |
ES-091-C |
|
ES-091-A (human) ES-092-A (rat) |
|
ES-091-M400UA |
| BB2 |
ES-090-C |
|
|
|
ES-090-M400UA |
| Calcitonin |
AM1 |
|
|
|
|
6110136400UA |
| AM2 |
ES-430-C |
ES-430-CF |
ES-430-A |
|
ES-430-M400UA |
| CGRP1 |
ES-420-C |
ES-420-CF |
ES-420-A |
ES-420-AF |
ES-420-M400UA (CHO-K1) 6110135400UA (SF9) RBHGRPM400UA (SK-N-MC) |
| Cannabinoid |
CB1 |
ES-110-C |
|
ES-110-A |
ES-110-AF |
ES-110-M400UA (CHO-K1) 6110129400UA (SF9) RBHCB1M400UA (HEK293) |
| CB2 |
ES-111-C (CHO-K1) RBXCB2C (HEK293) |
ES-111-CF |
|
|
ES-111-M400UA (CHO-K1) 6110130400UA (SF9) RBXCB2M400UA (HEK293) |
| Chemerin |
GPR1 |
|
|
ES-661-A |
ES-661-AF |
|
| Chemokine |
CCR1 |
ES-132-C (CHO-K1) RBHCC1C (HEK293) |
ES-132-CF |
|
|
RBHCC1M400UA |
| CCR2b |
ES-133-C |
|
ES-133A |
ES-133-AF |
ES-133-M400UA (CHO-K1) 6110550400UA (HEK293) |
| CCR3 |
ES-138-C |
|
ES-138A |
ES-138-AF |
ES-138-M400UA |
| CCR6 |
ES-139-C |
ES-139-CF |
ES-139A |
ES-139-AF |
ES-139-M400UA |
| CCR7 |
ES-140-C |
ES-140-CF |
ES-140A |
ES-140-AF |
ES-140-M400UA |
| CCR8 |
ES-136-C |
|
ES-136A |
ES-136-AF |
ES-136-M400UA |
| CCR9a |
|
|
ES-146A |
ES-146-AF |
|
| CCR10 |
|
|
ES-143A |
ES-143-AF |
|
| CX3CR1 |
ES-137-C |
|
ES-137A |
ES-137-AF |
ES-137-M400UA |
| CXCR2 |
ES-145-C |
ES-145-CF |
ES-145A |
ES-145-AF |
ES-145-M400UA (CHO-K1) 6110132400UA (SF9) |
| CXCR3 |
ES-142-C |
|
ES-142A |
ES-142-AF |
ES-142-M400UA |
| CXCR6 |
ES-170-C |
ES-170-C |
ES-170A |
ES-170-AF |
ES-720-M400UA (CHO-K1) RBHCX6M400UA (HEK293) |
| XCR1 |
ES-148-C |
|
ES-148A |
ES-148-AF |
ES-148-M400UA |
| Chemokine |
CCK1 |
ES-530-C |
|
ES-530-A |
|
ES-530-M400UA (1321N1) 6110125400UA (SF9)
6110508400UA (NIH-3T3) |
| CCK2 |
ES-531-C |
|
ES-531-A |
|
ES-531-M400UA (1321N1) RBHCKBM400UA (HEK293) |
| Corticotropin Releasing Factor |
CRF1 |
ES-152-C |
|
ES-152-A |
|
ES-152-M400UA (CHO-K1) RBHCRF1M400UA (HEK293) |
| Dopamine |
D1 |
ES-172-C (CHO-K1) MCL-505 (CH4CI) MCL-506 (L Cells) |
ES-172-CF |
|
|
ES-172-M400UA (CHO-K1) 6110513400UA (L Cells) |
| D2L |
|
|
ES-171-A |
ES-171-AF |
6110137400UA |
| D25 |
|
|
|
|
RBHD2CM400UA |
| D3 |
ES-173-C |
|
|
|
ES-173-M400UA (human) 6110139400UA (rat) |
| D4 |
ES-170-C |
|
|
|
|
| D4.2 |
|
|
|
|
RBHD42M400UA (CHO-K1) 6110112400UA (SF9) |
| D4.4 |
MCL-507 |
|
|
|
RBHD44M400UA (CHO-K1) 6110122400UA (SF9) |
| D4.7 |
|
|
|
|
RBHD47M400UA (CHO-K1) 6110123400UA (SF9) |
| Endothelin |
ETA |
ES-320-C |
|
ES-320-A |
ES-320-AF |
ES-320-M400UA |
| ETB |
ES-321-C |
|
ES-321-A |
ES-321-AF |
ES-321-M400UA |
| Formyl Peptide |
FPR2 (FPRL1) |
ES-610-C |
ES-610-CF |
ES-610-A |
ES-610-AF |
ES-610-M400UA |
| Free Fatty Acid |
FFA1 (GPR40) |
ES-652-C |
|
ES-652-A |
ES-652-AF |
|
| FFA1 (GPR120) |
|
|
ES-800-A |
ES-800-AF |
|
| GABAB |
GABAB1a |
|
|
|
|
6110545400UA (CHO-K1) 6110560400UA (HEK293) |
| GABAB1b |
|
|
|
|
6110546400UA (CHO-K1) 6110557400UA (HEK293) |
| GABAB1a/B2 |
ES-500-C |
ES-500-CF |
ES-500-A |
|
ES-500-M400UA (CHO-K1) 6110559400UA (HEK293) |
| Galanin |
GAL1 |
ES-510-C (CHO-K1)
MCL-513 (HEK293)
RBXGL1C (HEK293) |
ES-510-CF |
ES-510-A |
ES-510-AF |
ES-510-M400UA (CHO-K1) 6110537400UA (HEK293) |
| GAL2 |
ES-511-C |
|
ES-511-A AX-008-PCF |
ES-511-AF |
ES-511-M400UA |
| Ghrelin |
ghrelin |
ES-410-C |
|
ES-410-A |
ES-410-AF |
ES-410-M400UA (CHO-K1) RBHGHSM400UA (HEK293) |
| Glucagon |
glucagon |
ES-710-C |
|
ES-710-A |
|
|
| GIP |
|
|
|
|
RBHGIPM400UA |
| GLP-2 |
ES-711-C |
ES-711-CF |
|
|
|
| Secretin |
|
|
ES-712-A |
ES-712-AF |
|
| Glutamate |
mGlu5A |
|
|
|
|
ES-555-M400UA |
| mGlu7 |
ES-553-C |
ES-553-CF |
|
|
|
| Glycoprotein Hormone |
TSH |
|
|
ES-790-A |
|
|
| Gonadotropin-releasing Hormone |
GnRH |
|
|
ES-600-A |
|
ES-600-M400UA |
| GPR |
OXGR1 |
|
|
ES-743-A |
ES-743-AF |
|
| SUCNR1 (Succinate, GPR91) |
|
|
ES-744-A |
ES-744-AF |
|
| Histamine |
H1 |
ES-390-C |
|
ES-390-A |
ES-390-AF |
ES-390-M400UA |
| H2 |
ES-391-C |
ES-391-CF |
ES-391-A |
ES-391-AF |
ES-391-M400UA (CHO-K1 6110565400UA (HEK293) |
| H3 |
ES-392-C |
ES-392-CF |
ES-392-A |
ES-392-AF |
ES-392-M400UA |
| H4 |
ES-393-C |
|
ES-393-A |
ES-393-AF |
ES-393-M400UA |
| KiSS1 (Metastin) |
KiSS1 (GPR54) |
ES-630-C |
|
ES-630-A |
|
ES-630-M400UA (MDA-MB-435S) RBHMTSM400UA (CHO-K1) |
| Leukotriene |
BLT1(LTB4R1) |
ES-340-C |
ES-340-CF |
ES-340-A |
|
ES-340-M400UA |
| CysLT1 |
ES-470-C |
|
ES-470-A |
|
ES-470-M400UA |
| OXE (HM74-like) |
|
|
ES-640-A |
|
|
| Lysophospholipid |
S1P2 (EDG5) |
|
|
ES-594-A |
ES-594-AF |
|
| S1P4 (EDG6) |
|
|
ES-592-A |
ES-592-AF |
|
| S1P5 (EDG8) |
|
|
ES-593-A |
ES-593-AF |
|
| Mas related |
MrgX1 |
|
|
ES-740-A |
|
|
| MrgX2 |
|
|
ES-742-A |
|
|
| MrgB3 |
|
|
ES-745-A |
ES-745-AF |
|
| Melanin-Concentrating Hormone |
MCH1 |
ES-370-C |
|
ES-370-A |
ES-370-AF |
ES-370-M400UA |
| MCH2 |
ES-372-C |
|
ES-371-A |
ES-371-AF |
ES-372-M400UA |
| Melanocortin |
MC1 |
ES-195-C |
ES-195-CF |
|
|
ES-195-M400UA |
| MC3 |
ES-193-C (human) ES-190-C (mouse) |
ES-193-CF (human) ES-190-CF (mouse) |
|
|
ES-193-M400UA (human) RBXMC3M400UA (human) ES-190-M400UA (mouse) |
| MC4 |
ES-191-C |
ES-191-CF |
ES-191-A |
|
ES-191-M400UA (CHO-K1) RBHMC4M400UA (HEK293) |
| MC5 |
ES-194-C RBXMC5C ES-192-C |
ES-194-CF ES-192-CF |
|
|
ES-191-M400UA (human) RBXMC5M400UA (human) ES-192-M400UA (mouse) |
| Melanocortin |
MT1 |
ES-620-C |
|
ES-620-A |
ES-620-AF |
ES-620-M400UA |
| MT2 |
ES-621-C |
|
ES-621-A |
ES-621-AF |
ES-621-M400UA |
| Motilin |
motilin |
ES-380-C (CHO-K1) RBHMOTC (HEK293) |
|
ES-380-A |
|
ES-380-M400UA (CHO-K1) RBHMOTM400UA (HEK293) |
| Neuromedin U |
NMU1 |
ES-450-C |
|
ES-450-A |
|
ES-450-M400UA (CHO-K1) RBHNU1M400UA (HEK293) |
| NMU2 |
ES-451-C |
|
ES-451-A |
|
ES-451-M400UA (CHO-K1) RBHNU2M400UA (HEK293) |
| Neuropeptide S |
NPS |
ES-770-C |
|
ES-770-A |
|
|
| Neuropeptide FF |
NPFF1 |
ES-491-C |
ES-491-CF |
|
|
ES-491-M400UA (CHO-K1) RBHNF1M400UA (CHO-DHFR - ) |
| NPFF2 |
ES-490-C |
ES-490-CF |
ES-490-A |
|
RBHNF2M400UA |
| Neuropeptide W/B |
NPBW2 (GPR8) |
|
|
|
|
RBHGP8M400UA |
| Neuropeptide Y |
Y1 |
ES-351-C |
ES-351-CF |
ES-351-A |
|
6110133400UA (SF9) RBHNP1M400UA (SK-N-MC) |
| Y2 |
ES-352-C |
ES-352-CF |
ES-352-A |
|
RBHNP2M400UA |
| Neurotensin |
NTS1 |
ES-690-C RBXNT1C |
|
ES-690-A |
|
ES-690-M400UA (CHO-K1) 6110518400UA (CHO-K1) RBXNT1M400UA (HEK293) |
| NTS2 |
ES-691-C |
|
|
|
ES-691-M400UA (1321N1) 6110566400UA (HEK293) |
| Nicotinic |
GPR109A (HM74A) |
ES-760-C |
ES-760-CF |
ES-760-A |
|
ES-760-M400UA (CHO-K1) RBHNICM400UA (IMR32) |
| Opioid |
delta |
|
|
|
|
RBHODM400UA (human) 6110549400UA (human) 6110115400UA (mouse) |
| kappa |
ES-541-C |
|
ES-541-A |
|
ES-541-M400UA (CHO-K1) 6110558400UA (HEK293) |
| mu |
ES-542-C |
ES-542-CF |
ES-542-A |
ES-542-AF |
ES-542-M400UA |
| NOP (ORL1) |
ES-230-C (CHO-K1) RBHORLC (HEK293) |
ES-230-CF |
ES-230-A |
|
6110540400UA (CHO-K1) RBHORLM400UA (HEK293) |
| Orexin |
OX1 |
ES-330-C |
|
ES-330-A |
|
ES-330-M400UA |
| OX2 |
ES-331-C |
|
ES-331-A |
|
ES-331-M400UA |
| Peptide P518 |
QRFP (OX2-like, GPR103) |
ES-670-C |
|
ES-670-A |
|
ES-670-M400UA (CHO-K1) RBH103M400UA (HEK293) |
| Prokineticin |
PKR1 |
|
|
ES-750-A |
ES-750-A |
ES-750-M400UA |
| PKR2 |
ES-751-C |
ES-751-CF |
ES-751-A |
ES-751-AF |
ES-751-M400UA (CHO-K1) RBHPK2M400UA (HEK293) |
| Prolactin Releasing Peptid |
PRRP |
ES-480-C |
|
ES-480-A |
|
ES-480-M400UA |
| Prostanoid |
DP1 |
ES-560-C |
|
ES-560-A |
|
|
| DP2 (CRTH2) |
ES-561-C |
ES-561-CF |
ES-561-A |
|
ES-561-M400UA (CHO-K1) RBHTH2M400UA (HEK293) |
| EP2 |
ES-562-C |
ES-562-CF |
|
|
ES-562-M400UA |
| EP4 |
ES-563-C |
|
ES-563-A |
|
|
| FP |
ES-564-C |
|
|
|
|
| TP |
RBHTPC |
|
|
|
RBHTPM400UA |
| Protease-activated |
PAR2 |
|
|
ES-780-A |
|
|
| PAR4 |
|
|
ES-782-A |
ES-782-AF |
|
| Purinergic P2Y |
P2Y1 |
RBHP1C |
|
|
|
|
| P2Y2 |
ES-290-C |
|
|
|
|
| P2Y4 |
RBHP4C |
|
|
|
|
| P2Y6 |
ES-292-C |
|
|
|
|
| P2Y11 |
RBHP11C |
|
ES-293-A |
ES-293-AF |
|
| P2Y12 |
RBHP12C |
|
|
|
|
| Relaxin |
RXFP3 |
ES-656-C |
ES-656-CF |
ES-656-A |
|
ES-656-M400UA |
| RXFP4 |
ES-659-C |
|
ES-659-A |
|
ES-659-M400UA |
| Somatostatin |
sst1 |
ES-520-C |
|
|
|
ES-520-M400UA |
| sst2a |
ES-521-C |
ES-521-CF |
ES-521-A |
ES-521-AF |
ES-521-M400UA |
| sst3 |
ES-523-C |
ES-523-CF |
ES-523-A |
|
ES-523-M400UA |
| sst4 |
ES-524-C (CHO-K1)
RBHST4C (HEK293) |
ES-524-CF |
ES-524-A |
ES-524-AF |
ES-524-M400UA (CHO-K1) RBHST4M400UA (HEK293) |
| sst5 |
ES-522-C (CHO-K1) RBHST5C (HEK293) |
ES-522-CF |
ES-522-A |
Es-522-AF |
ES-522-M400UA (CHO-K1) RBHST5M400UA (HEK293) |
| Tachykinin |
NK1 |
|
|
|
|
6110551400UA |
| NK2 |
ES-251-C |
|
ES-251-A |
|
ES-251-M400UA |
| NK3 |
ES-252-C |
|
ES-252-A |
|
ES-252-M400UA |
| Thyrotropin Releasing Hormone |
TRH1 |
ES-700-C |
|
ES-700-A |
ES-700-AF |
ES-700-M400UA |
| Urotensin |
UT (Uro II, GPR14) |
ES-440-C |
|
ES-440-A (human) AX-007-PCF (human) ES-441-A (rat) |
ES-440-AF |
ES-440-M400UA (human) RBMUR2M400UA (mouse) |
| Vasoactive Intestinal Peptide |
PAC1 (PACAP) |
|
|
ES-272-A |
|
|
| VPAC1 (VIP) |
|
|
ES-273-A |
|
RBHVIPM400UA |
| VPAC2 |
|
|
ES-274-A |
|
|
| Vasopressin |
V1A |
ES-361-C |
|
ES-361-A |
ES-361-AF |
ES-361-M400UA (1321N1)
RBHV1AM400UA (HEK293) |
| V1B |
ES-362-C (human)
RBHV1BC (human)
ES-360-C (rat) |
|
ES-362-A |
ES-362-AF |
ES-362-M400UA (human)
RBHV1BM400UA (human) 6110543400UA (human) ES-360-M400UA (rat) |
| V2 |
ES-363-C |
ES-363-CF |
ES-363-A |
|
ES-363-M400UA (1321N1)
6110541400UA (CHO-K1) |